Target Details
| UniProt AC | Q8NBP7 |
|---|---|
| Gene Symbol | PCSK9 |
| Protein Name | Proprotein convertase subtilisin/kexin type 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05922 (Inhibitor_I9) PF18459 (PCSK9_C1) PF18464 (PCSK9_C2) PF18463 (PCSK9_C3) PF00082 (Peptidase_S8) |
Summary
- Multi-target molecules 227
- Clinical molecules 0
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (227)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VVFBDPKAWCMBFC
|
6.4 | IC50 | 2 | — | |
WEBMSJYTWXDLIP
|
6.4 | IC50 | 2 | — | |
BJBASKROIULEMR
|
6.4 | Ki | 2 | — | |
FSWBQPGSMBLQBY
|
6.4 | IC50 | 2 | — | |
RIMRVERSFDYITK
|
6.3 | IC50 | 2 | — | |
WDOZXDCBSSIRIX
|
6.3 | Ki | 2 | — | |
SUNSLACFIOGRFF
|
6.3 | IC50 | 2 | — | |
ALPNZVCVPJFQIU
|
6.3 | IC50 | 2 | — | |
AZFPODXRUNPZHM
|
6.3 | IC50 | 2 | — | |
BOEQQAQLLWKPTJ
|
6.3 | IC50 | 2 | — | |
BRBNSXUDJYDTAG
|
6.3 | IC50 | 2 | — | |
BTAAQTWWDLUMTF
|
6.3 | IC50 | 2 | — | |
CNGCIJQYBFMRMX
|
6.3 | IC50 | 2 | — | |
CRYTZKVYOZQLRR
|
6.3 | IC50 | 2 | — | |
CUHBJMSOISXVMR
|
6.3 | IC50 | 2 | — | |
DCPMQDCTYSJULX
|
6.3 | IC50 | 2 | — | |
DNZWZESQXUDNMY
|
6.3 | IC50 | 2 | — | |
DONIEJUKPWBLFP
|
6.3 | IC50 | 2 | — | |
DSUVELDKXDKGHU
|
6.3 | IC50 | 2 | — | |
FMNPUNYDOXDGJL
|
6.3 | IC50 | 2 | — | |
FOZMZJIMMVCKDE
|
6.3 | IC50 | 2 | — | |
FTHXTCAXAGRYFO
|
6.3 | IC50 | 2 | — | |
GJJNMAVROKHYBE
|
6.3 | IC50 | 2 | — | |
GNZYKGNQNCDUGS
|
6.3 | IC50 | 2 | — | |
GYDLBEUNRPUORD
|
6.3 | IC50 | 2 | — | |
GYRYVQSHMAAQKC
|
6.3 | IC50 | 2 | — | |
HJJJHFVYQDSEFZ
|
6.3 | IC50 | 2 | — | |
HMSVYVLLKIGLFT
|
6.3 | IC50 | 2 | — | |
HVRHTDCRQSHYOI
|
6.3 | IC50 | 2 | — | |
IJMDXLMQQXPEEX
|
6.3 | IC50 | 2 | — | |
JGLBVZXAFLSBCU
|
6.3 | IC50 | 2 | — | |
JRGJGUZUUUKIDC
|
6.3 | IC50 | 2 | — | |
KASDPFCBFIWJGE
|
6.3 | IC50 | 2 | — | |
KYENQZFDWAELLQ
|
6.3 | IC50 | 2 | — | |
LQNHCVGOZPMYOV
|
6.3 | IC50 | 2 | — | |
LTZLQMSMMBBVJA
|
6.3 | IC50 | 2 | — | |
LYMYTGOIKDBELY
|
6.3 | IC50 | 2 | — | |
MOYBXIHKSBVEGD
|
6.3 | IC50 | 2 | — | |
NNDLHUHLCVZCQG
|
6.3 | IC50 | 2 | — | |
NXAWESRPHOWAJS
|
6.3 | IC50 | 2 | — | |
OKDDJQPOHMWTNM
|
6.3 | IC50 | 2 | — | |
ORVGAHROAPZBAA
|
6.3 | IC50 | 2 | — | |
OSLDLYWXYKWSBN
|
6.3 | IC50 | 2 | — | |
PBFLCRPIXMRFSM
|
6.3 | IC50 | 2 | — | |
PRCZAYMEHYDTNS
|
6.3 | IC50 | 2 | — | |
PRMMNARWNYGQRR
|
6.3 | IC50 | 2 | — | |
QBEFLWKVIFFKMQ
|
6.3 | IC50 | 2 | — | |
QFEZLQHDFGWYBB
|
6.3 | IC50 | 2 | — | |
QKHPCEZOONLJGL
|
6.3 | IC50 | 2 | — | |
QSQIUHYDUXLSSG
|
6.3 | IC50 | 2 | — |