Target Details
UniProt ACQ8NBP7
Gene SymbolPCSK9
Protein NameProprotein convertase subtilisin/kexin type 9
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF05922 (Inhibitor_I9) PF18459 (PCSK9_C1) PF18464 (PCSK9_C2) PF18463 (PCSK9_C3) PF00082 (Peptidase_S8)
Summary
  • Multi-target molecules 227
  • Clinical molecules 0
  • Avg pChEMBL 6.86
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (227)
InChIKey pChEMBL Type Targets Clinical
MFZAHCDUXVQHDG 7.3 IC50 2
NHAKTDNLCUBYIO 7.3 IC50 2
NRRUCUBIKFVVTF 7.3 IC50 2
NRZSNKPBLRFRCO 7.3 IC50 2
OHMWYKRRPHNKAY 7.3 IC50 2
OOBXOHWMTQHGPZ 7.3 IC50 2
OTAKLFUVEQRFQC 7.3 IC50 2
OUHIHZKBZJHMKN 7.3 IC50 2
OUHIHZKBZJHMKN 7.3 IC50 2
PEFANKFLDJZTTE 7.3 IC50 2
PKLWPELHYNFFSC 7.3 IC50 2
PMMGPFKPCNXWKH 7.3 IC50 2
PQCJVPLQTYCXHG 7.3 IC50 2
PSNROLOZFCGPOO 7.3 IC50 2
QRIOCRNXOURWNI 7.3 IC50 2
RBWKHLPGHMYEBU 7.3 IC50 2
RZFKCVRKHPUZSA 7.3 IC50 2
SIUIJEXTVIHXRM 7.3 IC50 2
SREPCAPKCNETHI 7.3 IC50 2
SROMRSNBDIXBNC 7.3 IC50 2
SZGNJXJONFTTMZ 7.3 IC50 2
TVWRUGYHFKQXJI 7.3 IC50 2
UPZHBFNFWJCORK 7.3 IC50 2
UTPUESWLNFEKOJ 7.3 IC50 2
UYTBZWJKJSZDPS 7.3 IC50 2
VEBUCFXLBZQBKJ 7.3 IC50 2
VEEBNTLUXIEQDX 7.3 IC50 2
VEJNOLOAWWWCED 7.3 IC50 2
WKKAQOPQRBMISJ 7.3 IC50 2
WRPFBABRQIASOS 7.3 IC50 2
XBMWLWQWZMXFJE 7.3 IC50 2
XCIVVNWSQRGLMD 7.3 IC50 2
XJIUUGQYWJGRIR 7.3 IC50 2
XODWNXFGTNVYHB 7.3 IC50 2
XUATYLDPLNNZEX 7.3 IC50 2
YFTHABGMWCGOAK 7.3 IC50 2
ZDFSJIHCRYLAMT 7.3 IC50 2
ZQFZHVFJXFINPM 7.3 IC50 2
ZWPQEWXCTYEVJU 7.3 IC50 2
HGLMFBHBAMWYHY 7.2 Ki 2
UTOIMUBAPYEYBD 7.2 IC50 2
NSTFRFKCUDSCEN 7.2 Ki 2
AFTCBZMZKYOMRS 7.1 IC50 3
XZNCSFCXWWVUCW 7.0 Ki 2
PINVMNVLSVYQKP 7.0 Ki 2
KLPYFSFJVFMBJS 7.0 Ki 2
VORHKYQSFSQEEO 7.0 Ki 2
BDEUYEAHVFTURG 6.9 IC50 2
BEILGIKXQDGLEW 6.9 IC50 2
CTWNVUQVDCMLSE 6.9 IC50 2
2D structure