Target Details
| UniProt AC | Q8NBP7 |
|---|---|
| Gene Symbol | PCSK9 |
| Protein Name | Proprotein convertase subtilisin/kexin type 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05922 (Inhibitor_I9) PF18459 (PCSK9_C1) PF18464 (PCSK9_C2) PF18463 (PCSK9_C3) PF00082 (Peptidase_S8) |
Summary
- Multi-target molecules 227
- Clinical molecules 0
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (227)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MFZAHCDUXVQHDG
|
7.3 | IC50 | 2 | — | |
NHAKTDNLCUBYIO
|
7.3 | IC50 | 2 | — | |
NRRUCUBIKFVVTF
|
7.3 | IC50 | 2 | — | |
NRZSNKPBLRFRCO
|
7.3 | IC50 | 2 | — | |
OHMWYKRRPHNKAY
|
7.3 | IC50 | 2 | — | |
OOBXOHWMTQHGPZ
|
7.3 | IC50 | 2 | — | |
OTAKLFUVEQRFQC
|
7.3 | IC50 | 2 | — | |
OUHIHZKBZJHMKN
|
7.3 | IC50 | 2 | — | |
OUHIHZKBZJHMKN
|
7.3 | IC50 | 2 | — | |
PEFANKFLDJZTTE
|
7.3 | IC50 | 2 | — | |
PKLWPELHYNFFSC
|
7.3 | IC50 | 2 | — | |
PMMGPFKPCNXWKH
|
7.3 | IC50 | 2 | — | |
PQCJVPLQTYCXHG
|
7.3 | IC50 | 2 | — | |
PSNROLOZFCGPOO
|
7.3 | IC50 | 2 | — | |
QRIOCRNXOURWNI
|
7.3 | IC50 | 2 | — | |
RBWKHLPGHMYEBU
|
7.3 | IC50 | 2 | — | |
RZFKCVRKHPUZSA
|
7.3 | IC50 | 2 | — | |
SIUIJEXTVIHXRM
|
7.3 | IC50 | 2 | — | |
SREPCAPKCNETHI
|
7.3 | IC50 | 2 | — | |
SROMRSNBDIXBNC
|
7.3 | IC50 | 2 | — | |
SZGNJXJONFTTMZ
|
7.3 | IC50 | 2 | — | |
TVWRUGYHFKQXJI
|
7.3 | IC50 | 2 | — | |
UPZHBFNFWJCORK
|
7.3 | IC50 | 2 | — | |
UTPUESWLNFEKOJ
|
7.3 | IC50 | 2 | — | |
UYTBZWJKJSZDPS
|
7.3 | IC50 | 2 | — | |
VEBUCFXLBZQBKJ
|
7.3 | IC50 | 2 | — | |
VEEBNTLUXIEQDX
|
7.3 | IC50 | 2 | — | |
VEJNOLOAWWWCED
|
7.3 | IC50 | 2 | — | |
WKKAQOPQRBMISJ
|
7.3 | IC50 | 2 | — | |
WRPFBABRQIASOS
|
7.3 | IC50 | 2 | — | |
XBMWLWQWZMXFJE
|
7.3 | IC50 | 2 | — | |
XCIVVNWSQRGLMD
|
7.3 | IC50 | 2 | — | |
XJIUUGQYWJGRIR
|
7.3 | IC50 | 2 | — | |
XODWNXFGTNVYHB
|
7.3 | IC50 | 2 | — | |
XUATYLDPLNNZEX
|
7.3 | IC50 | 2 | — | |
YFTHABGMWCGOAK
|
7.3 | IC50 | 2 | — | |
ZDFSJIHCRYLAMT
|
7.3 | IC50 | 2 | — | |
ZQFZHVFJXFINPM
|
7.3 | IC50 | 2 | — | |
ZWPQEWXCTYEVJU
|
7.3 | IC50 | 2 | — | |
HGLMFBHBAMWYHY
|
7.2 | Ki | 2 | — | |
UTOIMUBAPYEYBD
|
7.2 | IC50 | 2 | — | |
NSTFRFKCUDSCEN
|
7.2 | Ki | 2 | — | |
AFTCBZMZKYOMRS
|
7.1 | IC50 | 3 | — | |
XZNCSFCXWWVUCW
|
7.0 | Ki | 2 | — | |
PINVMNVLSVYQKP
|
7.0 | Ki | 2 | — | |
KLPYFSFJVFMBJS
|
7.0 | Ki | 2 | — | |
VORHKYQSFSQEEO
|
7.0 | Ki | 2 | — | |
BDEUYEAHVFTURG
|
6.9 | IC50 | 2 | — | |
BEILGIKXQDGLEW
|
6.9 | IC50 | 2 | — | |
CTWNVUQVDCMLSE
|
6.9 | IC50 | 2 | — |