Target Details
| UniProt AC | Q8NBP7 |
|---|---|
| Gene Symbol | PCSK9 |
| Protein Name | Proprotein convertase subtilisin/kexin type 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05922 (Inhibitor_I9) PF18459 (PCSK9_C1) PF18464 (PCSK9_C2) PF18463 (PCSK9_C3) PF00082 (Peptidase_S8) |
Summary
- Multi-target molecules 227
- Clinical molecules 0
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (227)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CXYIZMOWQIOCCP
|
8.6 | Ki | 2 | — | |
AJCMEMYQDXJTLA
|
8.5 | IC50 | 2 | — | |
KKTRCZWTWYYSCY
|
8.5 | IC50 | 2 | — | |
MVKQIKVUJHXYFL
|
8.4 | Ki | 2 | — | |
PGYQBTHDSQHEAE
|
8.4 | Ki | 2 | — | |
GEYNSTBJBJHKBR
|
8.4 | Ki | 2 | — | |
MUNCMINBJLDFBS
|
8.2 | Ki | 2 | — | |
PYVKCKXGZHKWHI
|
8.2 | IC50 | 2 | — | |
PNXFQQVLICCBOG
|
8.1 | IC50 | 2 | — | |
WBHDYRHQHHLKQI
|
7.7 | IC50 | 2 | — | |
SXUMLHZCSVRHKE
|
7.6 | Ki | 2 | — | |
ZRUWDDBTCYFPLA
|
7.6 | Ki | 2 | — | |
OMZKYRSDRNYKAZ
|
7.5 | Ki | 2 | — | |
OTKKOUJLPCKSCD
|
7.4 | Ki | 2 | — | |
TZQCDWGPFXCCFJ
|
7.3 | Ki | 2 | — | |
ASTBLTXEDYOOHH
|
7.3 | IC50 | 2 | — | |
BFBKGIZCMYXWKP
|
7.3 | IC50 | 2 | — | |
BPABXCYDPRUTJP
|
7.3 | IC50 | 2 | — | |
BPDDXYVTWKHSPJ
|
7.3 | IC50 | 2 | — | |
BYCVINHSHUVRLH
|
7.3 | IC50 | 2 | — | |
CBNRIGHHWFOMTR
|
7.3 | IC50 | 2 | — | |
CMEDPZMTGNTTBQ
|
7.3 | IC50 | 2 | — | |
DAFOIRPOHRTCCU
|
7.3 | IC50 | 2 | — | |
DQNPOFYOPIYJIW
|
7.3 | IC50 | 2 | — | |
FAQXSFYHHVOERA
|
7.3 | IC50 | 2 | — | |
FIGHUWBUPINGCK
|
7.3 | IC50 | 2 | — | |
FIGQUGWNWAGSMX
|
7.3 | IC50 | 2 | — | |
FVSGRCFFDUJBSM
|
7.3 | IC50 | 2 | — | |
GHYVELVQBCQZAW
|
7.3 | IC50 | 2 | — | |
HJWRADTVRMRTCL
|
7.3 | IC50 | 2 | — | |
HSGRVVJDCMQDDO
|
7.3 | IC50 | 2 | — | |
HSVBNERTWMNCEC
|
7.3 | IC50 | 2 | — | |
HTZAUHJLSZVMER
|
7.3 | IC50 | 2 | — | |
HVQDJWFAGPSFHW
|
7.3 | IC50 | 2 | — | |
HZSDNSSEFWHOAM
|
7.3 | IC50 | 2 | — | |
IBHCNYFVFVJSNW
|
7.3 | IC50 | 2 | — | |
IIACQYHQRJCFAR
|
7.3 | IC50 | 2 | — | |
IMEFOOHITUHVKM
|
7.3 | IC50 | 2 | — | |
IOHQDPRJGZKIKP
|
7.3 | IC50 | 2 | — | |
ISQOVBPPZKQLLB
|
7.3 | IC50 | 2 | — | |
IVTNLJRCNTZRGT
|
7.3 | IC50 | 2 | — | |
JBUXHFKZMXLWCD
|
7.3 | IC50 | 2 | — | |
JGLBVZXAFLSBCU
|
7.3 | IC50 | 2 | — | |
JHYDAIUPBQLKHW
|
7.3 | IC50 | 2 | — | |
JQXBYNLOSRYECM
|
7.3 | IC50 | 2 | — | |
KDFJEZBQMMRKJX
|
7.3 | IC50 | 2 | — | |
KICTXGZKQYJVHU
|
7.3 | IC50 | 2 | — | |
KJNMWJFZUNTGKI
|
7.3 | IC50 | 2 | — | |
LBFGAFNKUVYELA
|
7.3 | IC50 | 2 | — | |
LPLOQDKAJJIQHJ
|
7.3 | IC50 | 2 | — |