Target Details
UniProt ACQ8NBP7
Gene SymbolPCSK9
Protein NameProprotein convertase subtilisin/kexin type 9
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF05922 (Inhibitor_I9) PF18459 (PCSK9_C1) PF18464 (PCSK9_C2) PF18463 (PCSK9_C3) PF00082 (Peptidase_S8)
Summary
  • Multi-target molecules 227
  • Clinical molecules 0
  • Avg pChEMBL 6.86
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (227)
InChIKey pChEMBL Type Targets Clinical
CXYIZMOWQIOCCP 8.6 Ki 2
AJCMEMYQDXJTLA 8.5 IC50 2
KKTRCZWTWYYSCY 8.5 IC50 2
MVKQIKVUJHXYFL 8.4 Ki 2
PGYQBTHDSQHEAE 8.4 Ki 2
GEYNSTBJBJHKBR 8.4 Ki 2
MUNCMINBJLDFBS 8.2 Ki 2
PYVKCKXGZHKWHI 8.2 IC50 2
PNXFQQVLICCBOG 8.1 IC50 2
WBHDYRHQHHLKQI 7.7 IC50 2
SXUMLHZCSVRHKE 7.6 Ki 2
ZRUWDDBTCYFPLA 7.6 Ki 2
OMZKYRSDRNYKAZ 7.5 Ki 2
OTKKOUJLPCKSCD 7.4 Ki 2
TZQCDWGPFXCCFJ 7.3 Ki 2
ASTBLTXEDYOOHH 7.3 IC50 2
BFBKGIZCMYXWKP 7.3 IC50 2
BPABXCYDPRUTJP 7.3 IC50 2
BPDDXYVTWKHSPJ 7.3 IC50 2
BYCVINHSHUVRLH 7.3 IC50 2
CBNRIGHHWFOMTR 7.3 IC50 2
CMEDPZMTGNTTBQ 7.3 IC50 2
DAFOIRPOHRTCCU 7.3 IC50 2
DQNPOFYOPIYJIW 7.3 IC50 2
FAQXSFYHHVOERA 7.3 IC50 2
FIGHUWBUPINGCK 7.3 IC50 2
FIGQUGWNWAGSMX 7.3 IC50 2
FVSGRCFFDUJBSM 7.3 IC50 2
GHYVELVQBCQZAW 7.3 IC50 2
HJWRADTVRMRTCL 7.3 IC50 2
HSGRVVJDCMQDDO 7.3 IC50 2
HSVBNERTWMNCEC 7.3 IC50 2
HTZAUHJLSZVMER 7.3 IC50 2
HVQDJWFAGPSFHW 7.3 IC50 2
HZSDNSSEFWHOAM 7.3 IC50 2
IBHCNYFVFVJSNW 7.3 IC50 2
IIACQYHQRJCFAR 7.3 IC50 2
IMEFOOHITUHVKM 7.3 IC50 2
IOHQDPRJGZKIKP 7.3 IC50 2
ISQOVBPPZKQLLB 7.3 IC50 2
IVTNLJRCNTZRGT 7.3 IC50 2
JBUXHFKZMXLWCD 7.3 IC50 2
JGLBVZXAFLSBCU 7.3 IC50 2
JHYDAIUPBQLKHW 7.3 IC50 2
JQXBYNLOSRYECM 7.3 IC50 2
KDFJEZBQMMRKJX 7.3 IC50 2
KICTXGZKQYJVHU 7.3 IC50 2
KJNMWJFZUNTGKI 7.3 IC50 2
LBFGAFNKUVYELA 7.3 IC50 2
LPLOQDKAJJIQHJ 7.3 IC50 2
2D structure