Target Details
| UniProt AC | Q8N5S9 |
|---|---|
| Gene Symbol | CAMKK1 |
| Protein Name | Calcium/calmodulin-dependent protein kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 40
- Clinical molecules 9
- Avg pChEMBL 7.14
KEGG Pathways (1)
Active Molecules (40)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
10.4 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
10.3 | Kd | 408 | — | |
NXSJMRCTGYTSTK
|
8.0 | Kd | 200 | — | |
XJIRZGFXJJLMOT
|
8.0 | IC50 | 2 | — | |
GFADNMXBCPZLOT
|
7.9 | IC50 | 2 | — | |
VAYOUJHNIZVWCA
|
7.9 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.8 | Kd | 170 | — | |
XQVVPGYIWAGRNI
|
7.7 | Kd | 34 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
LIZGTJPPOJGDHW
|
7.6 | IC50 | 2 | — | |
AYDMRHKXWFMUFF
|
7.6 | IC50 | 2 | — | |
GZYIVQMHOULGOR
|
7.5 | IC50 | 2 | — | |
WVSBGSNVCDAMCF
|
7.5 | IC50 | 4 | — | |
NWXLOTLDKWYYDP
|
7.3 | IC50 | 2 | — | |
BNYXRPMABDQJJR
|
7.3 | Kd | 5 | — | |
QQWUGDVOUVUTOY
|
7.3 | Kd | 231 | Yes | |
JCMKBZIPVJCSSW
|
7.3 | IC50 | 2 | — | |
OYONTEXKYJZFHA
|
7.2 | Kd | 69 | Yes | |
BIIVYFLTOXDAOV
|
7.1 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
7.1 | Kd | 82 | Yes | |
OXICLXLJBMPGTO
|
7.0 | IC50 | 5 | — | |
MYKOWOGZBMOVBJ
|
6.9 | IC50 | 9 | — | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 91 | Yes | |
QLMHELCDKYDUPA
|
6.7 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.7 | Kd | 191 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
CPATWHLHNLJLTB
|
6.6 | IC50 | 2 | — | |
UBVFQVJPQKNVPY
|
6.6 | IC50 | 2 | — | |
LIHGFLPDHFTNOG
|
6.4 | IC50 | 2 | — | |
OKIHVJIMTWMQNF
|
6.4 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
XZXHXSATPCNXJR
|
6.2 | Kd | 165 | Yes | |
ZZSBPGIGIUFJRA
|
6.1 | Kd | 46 | — | |
BPNUQXPIQBZCMR
|
6.1 | Kd | 83 | Yes | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
GZZXEPJJXLJJEJ
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |