Target Details
| UniProt AC | Q8N568 |
|---|---|
| Gene Symbol | DCLK2 |
| Protein Name | Serine/threonine-protein kinase DCLK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03607 (DCX) PF00069 (Pkinase) |
Summary
- Multi-target molecules 9
- Clinical molecules 3
- Avg pChEMBL 6.74
Active Molecules (9)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DDTPGANIPBKTNU
|
8.0 | Kd | 8 | — | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
KTEIFNKAUNYNJU
|
6.4 | Kd | 114 | — | |
HFNKQEVNSGCOJV
|
6.1 | Kd | 65 | — | |
JOOXLOJCABQBSG
|
6.1 | Kd | 139 | — | |
OUSFTKFNBAZUKL
|
6.0 | Kd | 58 | Yes | |
OYONTEXKYJZFHA
|
6.0 | Kd | 69 | Yes |