Target Details
| UniProt AC | Q8N4C8 |
|---|---|
| Gene Symbol | MINK1 |
| Protein Name | Misshapen-like kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 209
- Clinical molecules 21
- Avg pChEMBL 6.88
Active Molecules (209)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MFAQYJIYDMLAIM
|
6.7 | Kd | 130 | Yes | |
CLODUYRNZMIONW
|
6.7 | IC50 | 3 | — | |
DQPYZHUAILXFJI
|
6.7 | Ki | 27 | — | |
FLEAYYMORDPWAJ
|
6.7 | Ki | 90 | — | |
KRIUNPBAQZGFQA
|
6.7 | Ki | 76 | — | |
MHCPAORAYMTGCZ
|
6.7 | Ki | 37 | — | |
MZIOLOXGGOLJMJ
|
6.7 | Ki | 12 | — | |
QPORZABOFXPRHM
|
6.7 | Ki | 18 | — | |
XNWKXXIGSPPPBH
|
6.7 | Ki | 31 | — | |
XVUSMHCLFMFBQR
|
6.7 | IC50 | 3 | — | |
YEKVTSRZMPLPFK
|
6.7 | Ki | 17 | — | |
NXSJMRCTGYTSTK
|
6.6 | Kd | 200 | — | |
ADMFLILDQJSEIK
|
6.6 | Ki | 72 | — | |
CNTCGRJDUJEUDG
|
6.6 | Ki | 37 | — | |
HXHAJRMTJXHJJZ
|
6.6 | Ki | 52 | Yes | |
IAKGNUWZPSPEKU
|
6.6 | Ki | 19 | — | |
KCKXYZOBGBJZEG
|
6.6 | Ki | 36 | — | |
NZVDDFRUBIEKLV
|
6.6 | Ki | 20 | — | |
OYONTEXKYJZFHA
|
6.6 | Kd | 69 | Yes | |
UAQJVFADAYIBGC
|
6.6 | Ki | 23 | — | |
VAMDLIMJLAPZGX
|
6.6 | Ki | 10 | — | |
XBYVOPRDASFDMY
|
6.6 | Ki | 42 | — | |
XJJYJNMNYDNXNO
|
6.6 | Ki | 23 | — | |
ZGZVRPRSFXRGCF
|
6.6 | Ki | 76 | — | |
ZWVZORIKUNOTCS
|
6.6 | Ki | 69 | — | |
WCWUXEGQKLTGDX
|
6.5 | Kd | 22 | Yes | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
BJJHHKOPTKQUFQ
|
6.5 | Ki | 3 | — | |
KWRXWPRFIUJQBP
|
6.5 | Ki | 25 | — | |
LVECPYVAIBNSRV
|
6.5 | Ki | 33 | — | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
NLUPJKQOKWBWFC
|
6.5 | Ki | 69 | — | |
PNKALLUVKOKYHZ
|
6.5 | Ki | 32 | — | |
QONPPIZSNSSCSK
|
6.5 | Ki | 45 | Yes | |
ULHGAQSVFPOUDY
|
6.5 | Ki | 43 | — | |
VKBFHTIUXUCYRQ
|
6.5 | Ki | 66 | — | |
VUHZDNOPEVGHEO
|
6.5 | Ki | 29 | — | |
XHORJSJFHVABEA
|
6.5 | Ki | 49 | — | |
YUOWJICKAJQZLS
|
6.5 | Ki | 35 | — | |
ZYTFPHRVOZXPGZ
|
6.5 | Ki | 30 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
RKBYYWVZFBATHQ
|
6.5 | IC50 | 12 | — | |
ZYZUOYYVHYGMDE
|
6.5 | IC50 | 4 | — | |
DLWMVUDMPMKGEE
|
6.4 | Ki | 24 | — | |
GCZJQTRRJPRFIP
|
6.4 | Ki | 10 | — | |
GDYZFFBMSBDTAA
|
6.4 | Ki | 60 | — | |
NFMGZVPRGVERNN
|
6.4 | Ki | 44 | — | |
OEEGUWWPGAZRIJ
|
6.4 | Ki | 21 | — | |
PTVPBWWDGZSEAF
|
6.4 | Ki | 63 | — | |
RITAVMQDGBJQJZ
|
6.4 | Ki | 33 | — |