Target Details
| UniProt AC | Q8N4C8 |
|---|---|
| Gene Symbol | MINK1 |
| Protein Name | Misshapen-like kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 209
- Clinical molecules 21
- Avg pChEMBL 6.88
Active Molecules (209)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OADRBDVURCEKRP
|
7.4 | Ki | 44 | — | |
BPNUQXPIQBZCMR
|
7.3 | Ki | 60 | — | |
WPHKIQPVPYJNAX
|
7.3 | Ki | 81 | — | |
AUDNGNGLLRZLDR
|
7.2 | Ki | 33 | — | |
OWRXHGAFWZFFCW
|
7.2 | Ki | 113 | — | |
RJZDECGDCKOHBV
|
7.2 | Ki | 70 | — | |
UYGYYOIUVFMGKQ
|
7.2 | Ki | 30 | — | |
VXYDJXMHISGSDA
|
7.2 | Ki | 59 | — | |
CTNPALGJUAXMMC
|
7.2 | Kd | 151 | — | |
YUVLZPSSXDFUHH
|
7.2 | IC50 | 3 | — | |
OLUKILHGKRVDCT
|
7.1 | Ki | 44 | Yes | |
RWKDVIAVTRRJIR
|
7.1 | Ki | 23 | — | |
SKKRZILJUKYLJS
|
7.1 | Ki | 25 | — | |
WINHZLLDWRZWRT
|
7.1 | Ki | 66 | — | |
YDWMUCKJUNLURC
|
7.1 | Ki | 24 | — | |
GUBJNPWVIUFSTR
|
7.1 | Kd | 103 | — | |
XZXHXSATPCNXJR
|
7.1 | Kd | 165 | Yes | |
XHKFYFCKCXKVPO
|
7.0 | IC50 | 5 | — | |
BPNUQXPIQBZCMR
|
7.0 | Kd | 83 | Yes | |
CRKQBJZCCHKEGI
|
7.0 | Ki | 20 | — | |
DFMCXVONDDGQIY
|
7.0 | Ki | 66 | — | |
GCBJDOWIQHMCMR
|
7.0 | Ki | 84 | — | |
HEKAIDKUDLCBRU
|
7.0 | Ki | 20 | — | |
JSDGKSMNPHJDFK
|
7.0 | Ki | 35 | — | |
JZTOUVBEZONDKA
|
7.0 | Ki | 80 | — | |
KOZOJNNVQMRVIW
|
7.0 | Ki | 4 | — | |
LRZYYIZFBXFSJB
|
7.0 | Ki | 69 | — | |
MOHYPRXHKRXDSE
|
7.0 | IC50 | 8 | — | |
MULNSLQVKKUPJN
|
7.0 | Ki | 41 | — | |
XJSFDMGICAWQFS
|
7.0 | Ki | 60 | — | |
XOOAAYRIVATZNM
|
7.0 | Ki | 55 | — | |
MVCOAUNKQVWQHZ
|
7.0 | IC50 | 54 | Yes | |
YVQOYBIBWBAHKH
|
6.9 | IC50 | 12 | — | |
CHADTINFLWZSKR
|
6.9 | Ki | 26 | — | |
HOYRWTWZUFFACV
|
6.9 | Ki | 28 | — | |
KTWBYGUSEYSRND
|
6.9 | Ki | 28 | — | |
QKFXSCNWJZKJSJ
|
6.9 | Ki | 7 | — | |
XPHWIERLJBFPFV
|
6.9 | Ki | 69 | — | |
YMIJUBCSOKSFRU
|
6.9 | Ki | 87 | — | |
NGFGTMFVWSDFPS
|
6.8 | IC50 | 32 | — | |
ADLPKFFMGIJZIM
|
6.8 | Ki | 44 | — | |
CXBBWVXSZINRCS
|
6.8 | Ki | 41 | — | |
HSMUWLLZAZCLHF
|
6.8 | Ki | 25 | — | |
JTRNNNVASYCTLO
|
6.8 | Ki | 14 | — | |
OSVUGUHRKMMBSE
|
6.8 | Kd | 170 | — | |
RYYNGWLOYLRZLK
|
6.8 | Ki | 104 | — | |
SRONQUHCRFZABC
|
6.8 | Ki | 28 | — | |
TVUWQDLBEOZVOU
|
6.8 | Ki | 41 | — | |
XXSPHNFKLDJDAK
|
6.8 | Ki | 26 | — | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes |