Target Details
| UniProt AC | Q8N4C8 |
|---|---|
| Gene Symbol | MINK1 |
| Protein Name | Misshapen-like kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 209
- Clinical molecules 21
- Avg pChEMBL 6.88
Active Molecules (209)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
DPEXRCOBPACFOO
|
8.9 | Ki | 36 | — | |
BYWYWLKBKIJAAJ
|
8.9 | IC50 | 2 | — | |
FUMCKNCUEAQHCV
|
8.5 | Ki | 103 | — | |
UIARLYUEJFELEN
|
8.4 | Kd | 289 | Yes | |
OUJZYQBEFNDJQN
|
8.4 | Ki | 71 | — | |
UMTWTCVTRDYHQQ
|
8.4 | Ki | 56 | — | |
BGYVWFZMYBWCNY
|
8.3 | Ki | 30 | — | |
LYADGAGFYYXXIO
|
8.2 | IC50 | 82 | — | |
VGEXRDWWPSGZDH
|
8.2 | IC50 | 4 | — | |
LPILBMJJRGTKOQ
|
8.2 | Ki | 27 | — | |
MASJMHFQMYAPJR
|
8.2 | Ki | 41 | — | |
SMRWVXLSRJWVBF
|
8.2 | Ki | 25 | — | |
ZGGIYFOLDBTZIL
|
8.2 | Ki | 27 | — | |
ODPGGGTTYSGTGO
|
8.1 | Kd | 153 | — | |
CLEGDJQQHUTCOW
|
8.1 | Ki | 43 | — | |
KHPCIHZXOGHCLY
|
8.1 | IC50 | 3 | — | |
LSLPDHNUWRDOGC
|
8.1 | Ki | 25 | — | |
UBPYILGKFZZVDX
|
8.1 | IC50 | 130 | Yes | |
PIQCTGMSNWUMAF
|
8.0 | Kd | 137 | Yes | |
SLKCVFPEQGHNSI
|
8.0 | Ki | 29 | — | |
WVXNSAVVKYZVOE
|
8.0 | IC50 | 92 | — | |
LACOMQAWPSFXQC
|
7.9 | Ki | 27 | — | |
PUYIXDDMOUMMRR
|
7.9 | Ki | 27 | — | |
RFBPWKMQWSIPEO
|
7.9 | Ki | 28 | — | |
QNABDSWBQJKBHK
|
7.9 | IC50 | 45 | — | |
KHGPYYFCIAISBU
|
7.8 | Ki | 31 | — | |
LCHCSKHPVCDXAU
|
7.8 | Ki | 30 | — | |
IVRXNBXKWIJUQB
|
7.8 | Kd | 10 | — | |
OAVGBZOFDPFGPJ
|
7.7 | Kd | 42 | Yes | |
CHTMRWQLNNRRFJ
|
7.7 | Ki | 70 | — | |
PLHUMPJXRHMFFR
|
7.7 | Ki | 28 | — | |
WDARYLSSWBWVCU
|
7.7 | Ki | 49 | — | |
YFNWWNRZJGMDBR
|
7.7 | Kd | 35 | — | |
YWTBGJGMTBHQTM
|
7.7 | Ki | 65 | — | |
UEFCSGDOOJJXTN
|
7.7 | IC50 | 46 | — | |
KARJFNUGCLEZKM
|
7.6 | IC50 | 3 | — | |
KNACLJBHKVSTDL
|
7.6 | Ki | 40 | — | |
MCCCQFAOMZMZKE
|
7.6 | Ki | 52 | — | |
NJPWCTYVEJIQBM
|
7.6 | Ki | 72 | — | |
RBXYGQNZRVPDNB
|
7.6 | Ki | 34 | — | |
XFEKSSMJINNJSX
|
7.6 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
7.6 | Kd | 191 | — | |
JWNPDZNEKVCWMY
|
7.5 | Kd | 57 | Yes | |
WINHZLLDWRZWRT
|
7.5 | Kd | 201 | Yes | |
IFPPYSWJNWHOLQ
|
7.5 | Ki | 52 | Yes | |
XUFLBSMTYMFOQH
|
7.5 | Ki | 43 | — | |
ZKLJKKASNXVQBZ
|
7.5 | Ki | 27 | — | |
BSFNGHCTZDCQBF
|
7.4 | Ki | 93 | — | |
CNQGNADBGYCKKV
|
7.4 | Ki | 25 | — |