Target Details
| UniProt AC | Q8N1C3 |
|---|---|
| Gene Symbol | GABRG1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 7.66
KEGG Pathways (7)
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HGPFVUUTSFNGNR
|
6.7 | Ki | 18 | — | |
GMVMGIYPRPPNMB
|
6.7 | Ki | 16 | — | |
ZRKQHHNVLRRZFQ
|
6.7 | Ki | 16 | — | |
PTRPQDMPYNOBTR
|
6.7 | IC50 | 16 | — | |
DATCQVJMADOCRS
|
6.7 | IC50 | 16 | — | |
GXUSNZYZTBJMIT
|
6.7 | Ki | 16 | — | |
SINAJPKUKOSXOT
|
6.7 | IC50 | 16 | — | |
WFRRJMYHDPXXFB
|
6.7 | Ki | 16 | — | |
YWCLXVVWMQVKRF
|
6.7 | IC50 | 16 | — | |
CELFESKDAXZKDL
|
6.6 | IC50 | 16 | — | |
HXXGVDKGNHCARX
|
6.6 | IC50 | 16 | — | |
VMNYVCMDPUOQEL
|
6.6 | Ki | 16 | — | |
GXFWOMYQHNODFA
|
6.6 | IC50 | 16 | — | |
HOTHDLMXYUFPSZ
|
6.6 | IC50 | 16 | — | |
QQONDVXXMVPYIB
|
6.6 | Ki | 16 | — | |
GCNSLTKPBZQFJK
|
6.6 | IC50 | 16 | — | |
ODIZUHKZJZYZAL
|
6.6 | IC50 | 16 | — | |
RTMFRAUTYIKCRK
|
6.6 | Ki | 16 | — | |
WNDIDYSCZWXEJF
|
6.6 | Ki | 16 | — | |
LOBNIVNGRUTMOS
|
6.5 | IC50 | 16 | — | |
WRUTXEAYYQYJHO
|
6.5 | Ki | 16 | — | |
HJGRBNHROFTASJ
|
6.5 | IC50 | 16 | — | |
YHZXFRGWTKYPKS
|
6.5 | Ki | 16 | — | |
GAQCKHAXURZXGX
|
6.5 | IC50 | 16 | — | |
VEWLYIAEUXDQBW
|
6.5 | IC50 | 16 | — | |
GDVGLPNNOCDLLD
|
6.5 | IC50 | 16 | — | |
GEFDSAOHFGLQEZ
|
6.5 | Ki | 17 | — | |
WCTCMHZWHMFZFN
|
6.5 | Ki | 17 | — | |
DDSULWHSYUPHBK
|
6.5 | IC50 | 16 | — | |
XRWYYMUIIXMQBL
|
6.5 | IC50 | 16 | — | |
DAYQXLQRTQODQF
|
6.4 | Ki | 16 | — | |
DNCFKDLZZSXXJP
|
6.4 | IC50 | 16 | — | |
MUPIUJYENVWEKT
|
6.4 | IC50 | 16 | — | |
NQFQEBQBZXSXIX
|
6.4 | IC50 | 16 | — | |
VNFZCRPFALLSNM
|
6.4 | IC50 | 16 | — | |
SQPWTARSPNZNEI
|
6.4 | IC50 | 16 | — | |
QCSFXCHHKYXLHE
|
6.4 | Ki | 16 | — | |
YFEZLTPSCJWVHI
|
6.4 | Ki | 16 | — | |
YOJAHANNNITYMX
|
6.4 | Ki | 16 | — | |
ZLAPTIDQRXJQQL
|
6.4 | IC50 | 16 | — | |
AEPFXRGRJZMVIF
|
6.3 | Ki | 17 | — | |
JBTLCAMUYYCXTA
|
6.3 | IC50 | 16 | — | |
DKCNNHVHQYMVTO
|
6.3 | IC50 | 16 | — | |
BDGWCPYUERFMMY
|
6.3 | Ki | 16 | — | |
UMYWGMKUCZAQJO
|
6.3 | Ki | 16 | — | |
FNZFELZOBRBQJY
|
6.3 | IC50 | 16 | — | |
IGCSLIVTBUKKRS
|
6.3 | IC50 | 16 | — | |
SRJOCJYGOFTFLH
|
6.3 | Ki | 16 | — | |
IKDYRDIWKFJQTR
|
6.3 | IC50 | 16 | — | |
PZWMQJZDDYQYGN
|
6.3 | Ki | 16 | — |