Target Details
| UniProt AC | Q8N1C3 |
|---|---|
| Gene Symbol | GABRG1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 7.66
KEGG Pathways (7)
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OMQHFPMEAPEGTA
|
7.1 | Ki | 16 | — | |
AEYRTFCCYIWUJJ
|
7.1 | Ki | 16 | — | |
NFXAWQDTYKJJTD
|
7.1 | IC50 | 16 | — | |
JSRKYARWMIOKOB
|
7.0 | Ki | 16 | — | |
LWLYOXPDYPYNHH
|
7.0 | IC50 | 16 | — | |
SZSNAHWJFCIUBV
|
7.0 | IC50 | 17 | — | |
WUNJCJOCGLXHNU
|
7.0 | IC50 | 16 | — | |
GSNCQRDETZIWAE
|
7.0 | Ki | 16 | — | |
KWHWSXISOMCUPZ
|
7.0 | IC50 | 16 | — | |
VDAHGXKTABYDOQ
|
7.0 | Ki | 16 | — | |
XJSZCKCJAMOVEP
|
7.0 | IC50 | 16 | — | |
OWUSBEXUSSJSDZ
|
7.0 | IC50 | 16 | — | |
KQTMWRZAVOUNCI
|
7.0 | IC50 | 16 | — | |
IIDOALWZHDFUQF
|
7.0 | IC50 | 16 | — | |
FQDQLHDSVITISC
|
7.0 | IC50 | 16 | — | |
YEFFWDGMWBFKHL
|
7.0 | Ki | 16 | — | |
RMGFIVKKLZZKNY
|
7.0 | IC50 | 16 | — | |
XVRONCOEBFKZEW
|
7.0 | IC50 | 16 | — | |
NMMJOCVBNVTBNP
|
6.9 | Ki | 16 | — | |
GQXSRHIFUJLCSW
|
6.9 | Ki | 16 | — | |
JYXHNHBKWZQGLB
|
6.9 | Ki | 16 | — | |
HWOWPGLTTSFLOQ
|
6.9 | Ki | 16 | — | |
VFKHADGYGKHTDK
|
6.9 | IC50 | 16 | — | |
LHSWKUZVAZKLHJ
|
6.9 | IC50 | 16 | — | |
VFPUCBWBLOQFPU
|
6.9 | IC50 | 16 | — | |
YZBJLGYBBNTKKL
|
6.9 | IC50 | 16 | — | |
VHBFFQKBGNRLFZ
|
6.9 | Ki | 21 | — | |
ACPUCHLYONVNTK
|
6.9 | Ki | 16 | — | |
XYLGLGFZLQRDKD
|
6.9 | Ki | 16 | — | |
BIHMYZHWJAFHBO
|
6.8 | IC50 | 16 | — | |
KOTFZRCPKVQWPP
|
6.8 | Ki | 16 | — | |
XLKFCRQJPWBJNW
|
6.8 | IC50 | 16 | — | |
KTFRBKXLNKKPEA
|
6.8 | IC50 | 16 | — | |
DGWAMRKYNYINRJ
|
6.8 | IC50 | 16 | — | |
QQXJSYFEJVOQLZ
|
6.8 | IC50 | 16 | — | |
VGZQARXDBOOWBF
|
6.8 | Ki | 16 | — | |
JTQDBIFZWJTIIQ
|
6.8 | Ki | 16 | — | |
JXKAURVNHHPPND
|
6.8 | IC50 | 16 | — | |
RHARCGZTSJROQQ
|
6.8 | Ki | 16 | — | |
RLKPTPBBRCFHEK
|
6.8 | IC50 | 16 | — | |
BXKSCEUJEPDZBI
|
6.8 | Ki | 16 | — | |
STQWWORVIGBLOE
|
6.8 | Ki | 16 | — | |
XAXZXMJZHNVJEQ
|
6.8 | Ki | 16 | — | |
CGOOGLSJSVATGZ
|
6.8 | Ki | 16 | — | |
FLHRNVLCKMTQAP
|
6.8 | Ki | 17 | — | |
JQHJWKNJYLNAFL
|
6.8 | IC50 | 16 | — | |
XLKFCRQJPWBJNW
|
6.8 | IC50 | 16 | — | |
CGVJPQYHXQIFPE
|
6.7 | Ki | 16 | — | |
PGTVWKLGGCQMBR
|
6.7 | IC50 | 16 | — | |
QKZNNAUSAVZXNE
|
6.7 | Ki | 16 | — |