Target Details
| UniProt AC | Q8N1C3 |
|---|---|
| Gene Symbol | GABRG1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 7.66
KEGG Pathways (7)
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VQENDYBPFSSMNH
|
7.7 | IC50 | 16 | — | |
VREFGVBLTWBCJP
|
7.7 | Ki | 7 | — | |
ATJJCAREUNMTAU
|
7.7 | Ki | 2 | — | |
BYEKIJACVDAPTD
|
7.7 | Ki | 16 | — | |
LLAKESJIQFAQJA
|
7.7 | IC50 | 16 | — | |
FQDQLHDSVITISC
|
7.7 | IC50 | 16 | — | |
HKLYPSSDHPAOJM
|
7.7 | IC50 | 16 | — | |
KQQPWYMLATZBCF
|
7.7 | Ki | 2 | — | |
RSEMKXACIMVTQP
|
7.7 | Ki | 16 | — | |
WRDHNUVAWMYMJK
|
7.7 | IC50 | 16 | — | |
AURFZBICLPNKBZ
|
7.7 | IC50 | 16 | — | |
ZFLBRINMIQTFNB
|
7.7 | Ki | 18 | — | |
CJYPUCKDMBCYEH
|
7.6 | IC50 | 16 | — | |
LNPSYDJGQQETLB
|
7.6 | Ki | 16 | — | |
SHTOUNSWZVCSOU
|
7.6 | IC50 | 16 | — | |
TWQDMCPDTPVCQP
|
7.6 | IC50 | 16 | — | |
VHQCVUYEMJHQEX
|
7.6 | Ki | 16 | — | |
DMFKLCONGDUSKT
|
7.6 | Ki | 2 | — | |
FVEJOOHXPUFGSK
|
7.6 | Ki | 2 | — | |
INPWMTZRFFFMOA
|
7.6 | Ki | 2 | — | |
JHDNCJGODWCHES
|
7.6 | IC50 | 16 | — | |
LIXHLXZPUZQKCT
|
7.6 | IC50 | 16 | — | |
MBBOXTKOOFAZLI
|
7.6 | IC50 | 16 | — | |
PDOZRVXKPBQAJH
|
7.6 | IC50 | 16 | — | |
JWLCOGXPTWMMDY
|
7.6 | Ki | 16 | — | |
KBVJZOBCOIANOX
|
7.6 | Ki | 16 | — | |
KNJIPGCWYQXXPI
|
7.6 | Ki | 2 | — | |
KOMBGWPXIHBMLL
|
7.6 | IC50 | 16 | — | |
NHXHETTUSFLPHY
|
7.6 | Ki | 2 | — | |
OSHQANHMWJQRHB
|
7.6 | Ki | 16 | — | |
ULMKSNRBNFFOJQ
|
7.6 | Ki | 16 | — | |
ZWJGDMSWCKASII
|
7.6 | IC50 | 16 | — | |
HSUCRXNJMPDNOG
|
7.6 | IC50 | 16 | — | |
JNWDOTPNEZYWGO
|
7.6 | Ki | 16 | — | |
JAFQEKAQGSQGTM
|
7.6 | Ki | 16 | — | |
KQTMWRZAVOUNCI
|
7.6 | IC50 | 16 | — | |
VIEKPLVJCPXIIB
|
7.6 | IC50 | 16 | — | |
XLKKKDPUVUIHEL
|
7.6 | IC50 | 16 | — | |
ZSDPALDTMGRNKW
|
7.6 | Ki | 2 | — | |
GKHILVGVNGQMGS
|
7.5 | Ki | 2 | — | |
AANJEGNNNSDLGW
|
7.5 | Ki | 16 | — | |
IUVGMHPHSQSOGI
|
7.5 | Ki | 2 | — | |
WPJDKKSDGLIQQB
|
7.5 | Ki | 16 | — | |
DRCGHGOPCPUYAI
|
7.5 | IC50 | 16 | — | |
NKIYALPHXLYICR
|
7.5 | IC50 | 16 | — | |
BTCSSZJGUNDROE
|
7.5 | Ki | 23 | — | |
FOSOKBNWILBLSN
|
7.5 | Ki | 16 | — | |
KTFRBKXLNKKPEA
|
7.5 | IC50 | 16 | — | |
ACVGNKYJVGNLIL
|
7.5 | IC50 | 16 | — | |
SCAPGUIFNHZJLH
|
7.5 | IC50 | 16 | — |