Target Details
UniProt ACQ8N1C3
Gene SymbolGABRG1
Protein NameGamma-aminobutyric acid receptor subunit gamma-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 485
  • Clinical molecules 0
  • Avg pChEMBL 7.66
Top Co-occurrence Targets
Active Molecules (485)
InChIKey pChEMBL Type Targets Clinical
PKJGSRHYDOGGLB 8.0 Ki 17
ZJQHPWUVQPJPQT 8.0 IC50 17
DHZINDHXJITJQU 7.9 Ki 2
FCBLAIZVPBQHMO 7.9 Ki 2
FJLMOGVUSSSKEC 7.9 Ki 16
HGXDYOKZLZBFJW 7.9 Ki 2
LLAKESJIQFAQJA 7.9 IC50 16
UXRDTECAKSYGRM 7.9 Ki 2
CNVQMRWAJHEFGZ 7.9 Ki 16
OPMIQGMTRGXAQY 7.9 IC50 16
PLDDKFUCCWRCBG 7.9 Ki 2
UDARHNNVNUUUEB 7.9 Ki 2
VAARLVBAANTQOM 7.9 Ki 16
KGIVKXMZIJEMJQ 7.9 Ki 2
NLCBGONMLZXCDS 7.9 Ki 2
QANMGLSLKPATOE 7.9 Ki 2
RXBGGFMEZUKQME 7.9 Ki 2
HSEWUGOOPIEKBZ 7.9 IC50 16
XAMVDLCXXPEEEG 7.9 Ki 16
PCGLDGXLCXIRGT 7.9 Ki 2
RXBGGFMEZUKQME 7.9 Ki 2
YLRURIRIQRAQJJ 7.9 Ki 16
ARMIIMXWCNOAOC 7.9 Ki 2
BAGQLZQXEXAEAA 7.9 Ki 2
LURVKJAOOMWPMR 7.8 Ki 2
WAEXHEOACCAOSS 7.8 Ki 16
FHTNSYDGFUAOSS 7.8 Ki 2
PHAFJLAQYPGVOC 7.8 Ki 2
RQNGTQFJWSNXHS 7.8 Ki 2
IMMPJABTWMVMPJ 7.8 Ki 16
IQXJMMLNUIUGIQ 7.8 Ki 16
PNRLOCDAUHBIHX 7.8 IC50 16
CKZVPJOTELQSHC 7.8 IC50 16
CPWJDGKKDQPBKJ 7.8 Ki 2
QCHBQARHFYCDNV 7.8 IC50 16
REIWWVZOVOIYMD 7.8 Ki 2
ZFPVOBQMGRHOBJ 7.8 IC50 16
CMVRRVIUBQXVIK 7.8 Ki 2
JWZNKJCEYMWLHS 7.8 IC50 16
MEWGBPFYMUBENF 7.8 IC50 16
NAXZRUMPHRMRDF 7.8 IC50 16
VXOXRIDQOBACKW 7.8 Ki 16
ZWNZTSDJEOGSPF 7.8 Ki 2
UKTUKCYHGVTZRH 7.8 Ki 2
UYXLFIXVNVPFAS 7.8 Ki 2
YJYRFBZSNPRHKU 7.8 IC50 16
ZLQICIASTSXSFD 7.8 Ki 2
IATKEJBVROWZSN 7.7 Ki 2
QVBUOPGWPXUAHT 7.7 IC50 16
UIPGLQFPZVUUQW 7.7 Ki 16
2D structure