Target Details
UniProt ACQ8N1C3
Gene SymbolGABRG1
Protein NameGamma-aminobutyric acid receptor subunit gamma-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 485
  • Clinical molecules 0
  • Avg pChEMBL 7.66
Top Co-occurrence Targets
Active Molecules (485)
InChIKey pChEMBL Type Targets Clinical
IQZNYMVWZKDNQS 8.2 Ki 2
OKZDZISQRKZKRC 8.2 Ki 2
HWUMRCHENDXGOC 8.2 Ki 2
INZCBQSEJUQCIX 8.2 Ki 2
YUOOYQDBXTWPKL 8.2 Ki 16
OTQXKRRISJPTFS 8.2 IC50 16
WMCJJXHYPNOCMT 8.2 IC50 16
WYEOFGFJCZYTHC 8.2 Ki 2
ZRPUPUBWCXFOCY 8.2 Ki 16
ZYTWOBRUUCLPMR 8.2 Ki 2
FAHMQYRQDMWTRG 8.1 Ki 2
IDYXWWMDHPHNDU 8.1 Ki 2
KFRCPAXRUYFZQC 8.1 Ki 2
LPOYLZZUEKLEBW 8.1 Ki 2
QWZAWUIUHQADCS 8.1 Ki 2
BBQPVOQVHLCYFA 8.1 Ki 2
RMBCZRNLGKJEAK 8.1 Ki 2
FICZDYQNTMRYOG 8.1 Ki 2
KMYUMBZLLVOGAP 8.1 Ki 2
DKCAUMRZSZVJCP 8.1 Ki 16
IVGTVZGLPHBTJV 8.1 IC50 16
IVGTVZGLPHBTJV 8.1 IC50 16
QTZCODMFYAFKIE 8.1 Ki 2
QVIQGNJPFOVZBZ 8.1 Ki 16
YHNNMZUUFMJQQY 8.1 IC50 16
CPBKEZZAUBJVEY 8.1 Ki 2
HCSPQICLTPISJP 8.1 Ki 2
XHWVFLWDNDWXHW 8.1 Ki 2
ZMBXNSVOASWJOO 8.1 Ki 2
XGJLRKVQXMSBJW 8.1 IC50 16
YTFLGZYWUGHFRL 8.1 Ki 2
IZRMALPAWZXIHR 8.0 Ki 2
NRJWKUBEWAELQW 8.0 Ki 2
BTGRTTKTGRILMF 8.0 Ki 2
FTLMOIDJQCYEHM 8.0 Ki 2
SZAYALFNNDVKGO 8.0 Ki 2
KWPOKTUWXDCATM 8.0 IC50 16
XZUVYGZTGVSFPM 8.0 Ki 2
AAOVKJBEBIDNHE 8.0 IC50 16
HQJSGBKPXYZTRN 8.0 IC50 16
MBZNSAJBODIJCK 8.0 IC50 16
PWFUHHSGSJDKCU 8.0 IC50 16
AKOKEYRHKIETQQ 8.0 Ki 2
GTGXTIRVKZBCGT 8.0 Ki 2
DQOWOBNQAJJKEH 8.0 Ki 2
PIZYEZVMCVAKJF 8.0 Ki 2
DVKHCFDZNVGRQT 8.0 IC50 16
HFPZDEHIDKJZSN 8.0 Ki 16
LMJMBPXKXWIKQK 8.0 IC50 16
NNHRCSJWUBQYQV 8.0 IC50 16
2D structure