Target Details
UniProt ACQ8N1C3
Gene SymbolGABRG1
Protein NameGamma-aminobutyric acid receptor subunit gamma-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 485
  • Clinical molecules 0
  • Avg pChEMBL 7.66
Top Co-occurrence Targets
Active Molecules (485)
InChIKey pChEMBL Type Targets Clinical
MKNXZRAKHYWDOS 8.4 IC50 16
NTKWVYCGMNXXNM 8.4 Ki 2
SAVPBGVTWKUBOS 8.4 Ki 2
XQUJTESAXUTXNH 8.4 Ki 16
YOOKLJJRQNYLGH 8.4 Ki 2
IELTUHSCGWKNTD 8.4 Ki 2
OPOMKDUZWWHXCK 8.4 Ki 2
ZOEVKYRFHVGOOY 8.4 Ki 2
ISEATUPRORNMRO 8.3 Ki 2
KFJIZPKNMXRHEO 8.3 Ki 2
CYGBAIOJMMSNSX 8.3 Ki 2
RGLUZPFSHJVPPP 8.3 Ki 2
UDAPJVKQJQNWQL 8.3 Ki 2
YGKSPOBIXHTPMV 8.3 IC50 16
UGPCGLRXJCIGIY 8.3 Ki 2
ACMQMUZDLQDWTK 8.3 Ki 16
GOCZPCXRIJMRNR 8.3 Ki 16
NAPZANZEQXWANH 8.3 Ki 2
PHOATQSOBKATTD 8.3 Ki 16
PTRXPVDOTUGGHW 8.3 IC50 16
QWWODAPIEHJFQG 8.3 IC50 16
UYITUPHIEXJHKX 8.3 Ki 2
BNANSHHVRHDWHQ 8.3 Ki 2
DAPYUYZNPMJDNB 8.3 Ki 2
KUMNWRPRQLCGBZ 8.3 Ki 2
UDTZRZLWBNBNCX 8.3 Ki 2
YMDCFKGDSKTSDY 8.3 Ki 2
LFONXNFQWUEXIC 8.3 Ki 2
QCWSWDXAJBAYEA 8.3 Ki 2
LOLNCKZNZWWETB 8.3 Ki 2
ZWWZTFYQCITUTK 8.3 IC50 16
NTKWVYCGMNXXNM 8.2 Ki 2
UASVNRUAMGFBRL 8.2 Ki 2
VTWITWDVHKQWCL 8.2 Ki 2
RMMFOEVSBRAPQP 8.2 Ki 2
TXIWNLQFRATZFL 8.2 Ki 4
AMHLDWGDZHKVKW 8.2 Ki 2
BTLWEEGNXUJKKB 8.2 IC50 16
KDVOBKXBJSUGHB 8.2 Ki 2
KIVQXKXZISOGBE 8.2 Ki 17
LKTVCZVRYOFEAX 8.2 Ki 2
NKIYALPHXLYICR 8.2 IC50 16
VBEASATUUNKOCC 8.2 Ki 2
YUSWMAULDXZHPY 8.2 Ki 20
ZRRVSALMQDOQAX 8.2 Ki 16
DPBNSJBWFFXHJY 8.2 Ki 2
PHAFJLAQYPGVOC 8.2 Ki 2
BDISWVKOOATATE 8.2 Ki 16
AFQKQBVQNAFSCA 8.2 Ki 2
CFFHDCIRJSILAR 8.2 Ki 2
2D structure