Target Details
UniProt ACQ8N1C3
Gene SymbolGABRG1
Protein NameGamma-aminobutyric acid receptor subunit gamma-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 485
  • Clinical molecules 0
  • Avg pChEMBL 7.66
Top Co-occurrence Targets
Active Molecules (485)
InChIKey pChEMBL Type Targets Clinical
ZOCSXAVNDGMNBV 8.6 IC50 16
JLXGTZZEOOJFOH 8.6 Ki 2
VRIQRWQZIAEDLB 8.6 Ki 2
OWAIKGZBRPVIGC 8.6 Ki 2
VHUKNSIDUVPWBR 8.6 Ki 2
IZUFYFBJMFQQAV 8.6 Ki 2
KUMNWRPRQLCGBZ 8.6 Ki 2
ZJLHYXXAIHFWMN 8.6 Ki 2
QSOBDJYLKIXMJX 8.6 Ki 2
CHIFCDOIPRCHCF 8.6 IC50 16
CHQPOBHNDRMXFK 8.6 Ki 18
COKVKKSOZBQKSG 8.5 Ki 2
ISYJVUADIFBVQO 8.5 Ki 2
LUUMGXGNVMPSEU 8.5 Ki 2
COFOXGPFFPFDIE 8.5 Ki 2
FNXCSTGZJQDVJJ 8.5 Ki 2
KVKYGVOAHGNAKZ 8.5 IC50 17
LENHHZQGSWCZJW 8.5 Ki 16
LPAODQAWVMEXKR 8.5 IC50 16
LSOGSCJAJAAADN 8.5 Ki 2
NEOUOHDNZDRDNJ 8.5 IC50 16
QIZPCEVRKTWHIE 8.5 IC50 16
RYLDZJANGRBUGW 8.5 IC50 16
DJLFGFRHHCQJCO 8.5 Ki 2
MXUSCXPVOCAUMX 8.5 Ki 2
NVRZICQXMRMPGV 8.5 Ki 2
ZMGVJHPLOILGKH 8.5 Ki 2
ABTNVOCRBNFBHY 8.5 Ki 2
XDRLVLSTZNMYLB 8.5 Ki 2
MVBVNOZDVRVMNH 8.4 IC50 16
VGKZDCNKIZAJPG 8.4 Ki 2
FCKVAABCJRWYHI 8.4 Ki 2
JLLCYCAJCAQIHF 8.4 Ki 2
RAKFVWDVZYUQCI 8.4 Ki 2
IEXRFFQPFNOGAP 8.4 Ki 2
SFMVPQDIOHQZIK 8.4 Ki 2
CBBFXXVRQALAPG 8.4 Ki 2
IZQOSQCYDUORJW 8.4 Ki 2
SRNKTNDYXGQRST 8.4 Ki 2
ACUNYYFYYWOKOD 8.4 IC50 16
AXPGZURVLRWNBR 8.4 Ki 16
BZVWONIGXAYZIT 8.4 IC50 16
CDWXZILKRXSANI 8.4 IC50 16
DYSDYZCGZCYPCT 8.4 IC50 16
JTYYMOMTGZSRFM 8.4 IC50 16
LMXUGQJMQSMLIQ 8.4 Ki 17
OJKALFLWJGRIRN 8.4 Ki 2
UFTKNTUWDMJOIX 8.4 IC50 16
UULFOYXSWNADTF 8.4 IC50 16
WOQHIJSDFJSXHI 8.4 Ki 2
2D structure