Target Details
| UniProt AC | Q8N1C3 |
|---|---|
| Gene Symbol | GABRG1 |
| Protein Name | Gamma-aminobutyric acid receptor subunit gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 485
- Clinical molecules 0
- Avg pChEMBL 7.66
KEGG Pathways (7)
Active Molecules (485)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZFKWSFOAVBLQM
|
9.8 | IC50 | 16 | — | |
WFPXOWCKXUEKCA
|
9.7 | IC50 | 16 | — | |
KVKWRJDNIJTMGN
|
9.6 | IC50 | 16 | — | |
QUUNMICPMYIHFS
|
9.4 | IC50 | 16 | — | |
VMDUABMKBUKKPG
|
9.4 | IC50 | 16 | — | |
XKENJWNGLCKOBP
|
9.3 | IC50 | 16 | — | |
NJUMMJUUDUYSKB
|
9.3 | IC50 | 16 | — | |
ALBKMJDFBZVHAK
|
9.3 | IC50 | 16 | — | |
BYMDBFGHCDTBMT
|
9.3 | IC50 | 16 | — | |
IUHKSTINHDUYRO
|
9.3 | IC50 | 16 | — | |
VJVAWKPXJCDEQG
|
9.3 | IC50 | 16 | — | |
WRXDVVALWQGPMW
|
9.3 | IC50 | 16 | — | |
ZNHJNGABIOBVSL
|
9.3 | Ki | 2 | — | |
BLJPKQXXDFIIFR
|
9.2 | IC50 | 16 | — | |
XJMIBNLJFYSGAR
|
9.2 | IC50 | 16 | — | |
JFGUJXZLJIUVPZ
|
9.1 | IC50 | 16 | — | |
LYFROTHEKIFZAU
|
9.1 | IC50 | 16 | — | |
RYIVVNHBYBYXHF
|
9.1 | IC50 | 16 | — | |
VZKRZUPJCVFVGR
|
9.1 | IC50 | 16 | — | |
DGBIGWXXNGSACT
|
9.1 | Ki | 16 | — | |
OFBIFZUFASYYRE
|
9.1 | Ki | 16 | — | |
YJZGQBGGTBIAOP
|
9.1 | IC50 | 16 | — | |
JSEPJHYIUICRFD
|
9.0 | Ki | 2 | — | |
AQKFCEWRKDXGMK
|
9.0 | Ki | 16 | — | |
FVFFDKKTXYVCCW
|
9.0 | IC50 | 16 | — | |
IPHSQMSRIWZULE
|
9.0 | Ki | 16 | — | |
KDMMIKQMHNBKAV
|
9.0 | Ki | 17 | — | |
KOVRZNUMIKACTB
|
9.0 | IC50 | 17 | — | |
LXQGNWWMMCBHEW
|
9.0 | Ki | 2 | — | |
RLFKILXOLJVUNF
|
9.0 | IC50 | 16 | — | |
WGRVAGIQTHEEQW
|
9.0 | IC50 | 16 | — | |
BSBLYLUAUVTSMM
|
9.0 | IC50 | 16 | — | |
VVCKCOBSJPEUNF
|
8.9 | Ki | 2 | — | |
NZBYBIYUIBGUGN
|
8.9 | Ki | 2 | — | |
LQBFIYUKUNNYLL
|
8.8 | Ki | 2 | — | |
CTFJMLYREQLXDJ
|
8.8 | Ki | 2 | — | |
RHGALLXQCYCOFY
|
8.8 | Ki | 2 | — | |
UIANKUAHFCTBLR
|
8.8 | Ki | 2 | — | |
OJLYUGSSUKAWJC
|
8.8 | Ki | 16 | — | |
ARLPBUKOJFUUPW
|
8.8 | Ki | 2 | — | |
MKFQRZJYNRVPBH
|
8.8 | Ki | 2 | — | |
KVKYGVOAHGNAKZ
|
8.7 | IC50 | 16 | — | |
MJTBJNQOWBQCJE
|
8.7 | Ki | 2 | — | |
OCZOXZDVTVVPSN
|
8.7 | Ki | 2 | — | |
FMAFUZDTDPMPLI
|
8.7 | Ki | 2 | — | |
ZQZXBWMDLMNNQJ
|
8.7 | Ki | 2 | — | |
YVURNXWPVAMMDF
|
8.7 | Ki | 2 | — | |
QTEUJQNPMLXVLL
|
8.7 | IC50 | 16 | — | |
UKHFPVCOXBJPIN
|
8.7 | IC50 | 17 | — | |
PAGIUELYHAPFIM
|
8.6 | Ki | 2 | — |