Target Details
UniProt ACQ8N1C3
Gene SymbolGABRG1
Protein NameGamma-aminobutyric acid receptor subunit gamma-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 485
  • Clinical molecules 0
  • Avg pChEMBL 7.66
Top Co-occurrence Targets
Active Molecules (485)
InChIKey pChEMBL Type Targets Clinical
MZFKWSFOAVBLQM 9.8 IC50 16
WFPXOWCKXUEKCA 9.7 IC50 16
KVKWRJDNIJTMGN 9.6 IC50 16
QUUNMICPMYIHFS 9.4 IC50 16
VMDUABMKBUKKPG 9.4 IC50 16
XKENJWNGLCKOBP 9.3 IC50 16
NJUMMJUUDUYSKB 9.3 IC50 16
ALBKMJDFBZVHAK 9.3 IC50 16
BYMDBFGHCDTBMT 9.3 IC50 16
IUHKSTINHDUYRO 9.3 IC50 16
VJVAWKPXJCDEQG 9.3 IC50 16
WRXDVVALWQGPMW 9.3 IC50 16
ZNHJNGABIOBVSL 9.3 Ki 2
BLJPKQXXDFIIFR 9.2 IC50 16
XJMIBNLJFYSGAR 9.2 IC50 16
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
VZKRZUPJCVFVGR 9.1 IC50 16
DGBIGWXXNGSACT 9.1 Ki 16
OFBIFZUFASYYRE 9.1 Ki 16
YJZGQBGGTBIAOP 9.1 IC50 16
JSEPJHYIUICRFD 9.0 Ki 2
AQKFCEWRKDXGMK 9.0 Ki 16
FVFFDKKTXYVCCW 9.0 IC50 16
IPHSQMSRIWZULE 9.0 Ki 16
KDMMIKQMHNBKAV 9.0 Ki 17
KOVRZNUMIKACTB 9.0 IC50 17
LXQGNWWMMCBHEW 9.0 Ki 2
RLFKILXOLJVUNF 9.0 IC50 16
WGRVAGIQTHEEQW 9.0 IC50 16
BSBLYLUAUVTSMM 9.0 IC50 16
VVCKCOBSJPEUNF 8.9 Ki 2
NZBYBIYUIBGUGN 8.9 Ki 2
LQBFIYUKUNNYLL 8.8 Ki 2
CTFJMLYREQLXDJ 8.8 Ki 2
RHGALLXQCYCOFY 8.8 Ki 2
UIANKUAHFCTBLR 8.8 Ki 2
OJLYUGSSUKAWJC 8.8 Ki 16
ARLPBUKOJFUUPW 8.8 Ki 2
MKFQRZJYNRVPBH 8.8 Ki 2
KVKYGVOAHGNAKZ 8.7 IC50 16
MJTBJNQOWBQCJE 8.7 Ki 2
OCZOXZDVTVVPSN 8.7 Ki 2
FMAFUZDTDPMPLI 8.7 Ki 2
ZQZXBWMDLMNNQJ 8.7 Ki 2
YVURNXWPVAMMDF 8.7 Ki 2
QTEUJQNPMLXVLL 8.7 IC50 16
UKHFPVCOXBJPIN 8.7 IC50 17
PAGIUELYHAPFIM 8.6 Ki 2
2D structure