Target Details
| UniProt AC | Q8N122 |
|---|---|
| Gene Symbol | RPTOR |
| Protein Name | Regulatory-associated protein of mTOR |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02985 (HEAT) PF14538 (Raptor_N) PF00400 (WD40) |
Summary
- Multi-target molecules 189
- Clinical molecules 3
- Avg pChEMBL 7.77
KEGG Pathways (12)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXCAKZGNKOZXBM
|
7.5 | IC50 | 7 | — | |
JWOWVKFLHKSOPE
|
7.5 | IC50 | 5 | — | |
UFKLYTOEMRFKAD
|
7.5 | IC50 | 6 | — | |
WXUZDBRGJSWGID
|
7.5 | IC50 | 5 | — | |
MFAQYJIYDMLAIM
|
7.5 | IC50 | 130 | Yes | |
BJEPBULKEVIYBP
|
7.5 | IC50 | 6 | — | |
FAUUWGBRPQXEOZ
|
7.5 | IC50 | 3 | — | |
LGAJJTHJWVAHRF
|
7.4 | IC50 | 6 | — | |
SWHLSVQEFGEDKB
|
7.4 | IC50 | 5 | — | |
XYFXUNWLLFSAGS
|
7.4 | IC50 | 5 | — | |
JOGKUKXHTYWRGZ
|
7.4 | IC50 | 28 | — | |
PYBNTHVXUJFNOG
|
7.4 | IC50 | 3 | — | |
CSLVGODBTQVCKU
|
7.3 | IC50 | 5 | — | |
VYGVLHBRKJFFMR
|
7.3 | IC50 | 5 | — | |
BFWNUTHNJXXPSV
|
7.3 | IC50 | 5 | — | |
TVISMJDQTRLBBY
|
7.3 | IC50 | 5 | — | |
RGGGKLOHVQCLKI
|
7.3 | IC50 | 3 | — | |
SXJWIRIRCLXOIF
|
7.3 | IC50 | 3 | — | |
QDNFQHRZXWGYKH
|
7.3 | IC50 | 8 | — | |
KUZSBKJSGSKPJH
|
7.2 | IC50 | 5 | — | |
WCTBFLLLNSMNGQ
|
7.2 | IC50 | 6 | — | |
FFFOZOQSDJISHN
|
7.2 | IC50 | 6 | — | |
LVGNJTOYOJYFMW
|
7.2 | IC50 | 3 | — | |
WLHXVOYGBREFJO
|
7.2 | IC50 | 6 | — | |
LBQBMEVXMVNFHK
|
7.2 | IC50 | 3 | — | |
NFISZJMWQXGLIR
|
7.2 | IC50 | 4 | — | |
SYKBZXMKAPICSO
|
7.2 | IC50 | 7 | — | |
LGWACEZVCMBSKW
|
7.2 | Ki | 7 | — | |
VZVYLEDIUUZTCW
|
7.2 | IC50 | 6 | — | |
BSJSHEXWIGDLOO
|
7.1 | IC50 | 6 | — | |
YWFOHQFLGQVFIB
|
7.1 | IC50 | 9 | — | |
TXZDQMGQQGAAGN
|
7.1 | IC50 | 5 | — | |
WZAQTKRFGGBJAQ
|
7.1 | IC50 | 3 | — | |
WLQPHPRJRBGPBN
|
7.1 | IC50 | 3 | — | |
WZDNUCMFYNAXQT
|
7.1 | IC50 | 4 | — | |
AHTXWEHJMLNLGH
|
7.1 | IC50 | 3 | — | |
NVRXTLZYXZNATH
|
7.1 | IC50 | 47 | Yes | |
UGDKPWVVBKHRDK
|
7.1 | IC50 | 6 | — | |
YMPHJTSPBGJDAR
|
7.0 | IC50 | 6 | — | |
QABQGNKUVHFGFL
|
7.0 | IC50 | 7 | — | |
WLHXVOYGBREFJO
|
7.0 | IC50 | 6 | — | |
BUOZDMLNVZSXNY
|
7.0 | IC50 | 3 | — | |
XRWVHPKHEAIWOF
|
7.0 | IC50 | 3 | — | |
ZLCNPQUYKAHNGY
|
7.0 | IC50 | 3 | — | |
DZIVLAHVAHIFES
|
7.0 | IC50 | 3 | — | |
ZTXMWXWZYOHCDZ
|
7.0 | IC50 | 3 | — | |
RBLRRVZXUXIHNG
|
7.0 | IC50 | 3 | — | |
BSJSHEXWIGDLOO
|
6.9 | IC50 | 6 | — | |
XXVSQSOIIVGFNA
|
6.9 | IC50 | 4 | — | |
XGLUOINQAVYTEU
|
6.9 | IC50 | 5 | — |