Target Details
| UniProt AC | Q8N122 |
|---|---|
| Gene Symbol | RPTOR |
| Protein Name | Regulatory-associated protein of mTOR |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02985 (HEAT) PF14538 (Raptor_N) PF00400 (WD40) |
Summary
- Multi-target molecules 189
- Clinical molecules 3
- Avg pChEMBL 7.77
KEGG Pathways (12)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IMXHGCRIEAKIBU
|
8.3 | IC50 | 5 | — | |
BIYXBMJPSRSLCH
|
8.2 | IC50 | 3 | — | |
OYXPDKVBMCFEJF
|
8.2 | IC50 | 5 | — | |
AWOSFEUBLOFLFP
|
8.2 | IC50 | 6 | — | |
RGOBXIPHRILFRR
|
8.2 | IC50 | 5 | — | |
KHRNSXIHUJHLRG
|
8.1 | IC50 | 3 | — | |
UHBBECJRCILYHF
|
8.1 | IC50 | 3 | — | |
WLQPHPRJRBGPBN
|
8.1 | IC50 | 3 | — | |
VLSSMLSPCKXABU
|
8.1 | IC50 | 4 | — | |
WGYPOAXANMFHMT
|
8.1 | IC50 | 10 | Yes | |
YDFGZXSSYDSJRM
|
8.1 | IC50 | 6 | — | |
AQODXCHGIFZIIO
|
8.1 | IC50 | 3 | — | |
KYHDRKVDXZQWIA
|
8.1 | IC50 | 3 | — | |
CEPOCJCCKQHPAE
|
8.1 | IC50 | 5 | — | |
FFGUSRSMWFYKGK
|
8.1 | IC50 | 5 | — | |
WQBAZXIQANTUOY
|
8.0 | IC50 | 4 | — | |
BMXAXHINKBUJQZ
|
8.0 | IC50 | 3 | — | |
BQSHYPCVOOBERM
|
8.0 | IC50 | 3 | — | |
CSTRZYJUXMVMTK
|
8.0 | IC50 | 3 | — | |
DVKYZVMXIFFGCQ
|
8.0 | IC50 | 3 | — | |
IEEJBCKDNGRROT
|
8.0 | IC50 | 3 | — | |
IJKMMCIUUSMYJP
|
8.0 | IC50 | 3 | — | |
IXGXFXPKQGUFLV
|
8.0 | IC50 | 3 | — | |
JAIMBGXDCZXCJM
|
8.0 | IC50 | 3 | — | |
LQOZCVYFWINNKE
|
8.0 | IC50 | 3 | — | |
NPZGBXGMPLHOLI
|
8.0 | IC50 | 3 | — | |
NVSABGFUPYOXBC
|
8.0 | IC50 | 3 | — | |
PORABIULAYKSHM
|
8.0 | IC50 | 3 | — | |
RFSMUFRPPYDYRD
|
8.0 | IC50 | 5 | — | |
YBVDOWOAPVPVJA
|
8.0 | IC50 | 3 | — | |
YKMDFLBFXDXLSC
|
8.0 | IC50 | 3 | — | |
YLDJDXDYJDCIEK
|
8.0 | IC50 | 3 | — | |
YTQAUCZNPTYTRY
|
8.0 | IC50 | 3 | — | |
YXNXKPZWTPLWQK
|
8.0 | IC50 | 3 | — | |
BIYXBMJPSRSLCH
|
7.9 | IC50 | 3 | — | |
IZLPVLBNRGPOHA
|
7.8 | IC50 | 5 | — | |
QUBPAMUWIHBFNS
|
7.8 | IC50 | 3 | — | |
GSZOKDIAJHWSJC
|
7.8 | IC50 | 3 | — | |
JYSGBOOAYHHKRU
|
7.8 | IC50 | 3 | — | |
KYHDRKVDXZQWIA
|
7.8 | IC50 | 3 | — | |
BHQVZJBRLXMAGL
|
7.7 | IC50 | 3 | — | |
MLNSAGOBCFMEKI
|
7.7 | IC50 | 6 | — | |
DXYGEHPPAYSYLJ
|
7.7 | IC50 | 3 | — | |
TUVCWJQQGGETHL
|
7.7 | IC50 | 22 | — | |
AKKCGLXULFRAET
|
7.7 | Ki | 7 | — | |
JROFGZPOBKIAEW
|
7.7 | IC50 | 10 | — | |
LFGXKIVXIWOATF
|
7.7 | IC50 | 5 | — | |
GMYLVKUGJMYTFB
|
7.6 | IC50 | 7 | — | |
NDQIDSZBEUKRAW
|
7.6 | IC50 | 3 | — | |
KVEPKTYZFVUHKX
|
7.6 | IC50 | 3 | — |