Target Details
| UniProt AC | Q8MMZ7 |
|---|---|
| Gene Symbol | PKG |
| Protein Name | cGMP-dependent protein kinase |
| Organism | Toxoplasma gondii |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00027 (cNMP_binding) PF00069 (Pkinase) |
Summary
- Multi-target molecules 102
- Clinical molecules 7
- Avg pChEMBL 7.58
Active Molecules (102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OZTUULYOGSAFBT
|
7.7 | IC50 | 3 | — | |
HGALDAPNHYJZAJ
|
7.6 | IC50 | 11 | Yes | |
MZPILEJBIWMIFA
|
7.6 | IC50 | 3 | — | |
GDQXJQSQYMMKRA
|
7.5 | IC50 | 15 | — | |
BSGWEWBSWAVORO
|
7.4 | IC50 | 5 | — | |
CJFWNLXLAAHQJY
|
7.4 | IC50 | 11 | Yes | |
DUPSNQFPAJUAKA
|
7.4 | IC50 | 9 | Yes | |
NLZUZMDQCFLSME
|
7.4 | IC50 | 4 | — | |
KAEFKAWNHDHBCY
|
7.4 | IC50 | 3 | — | |
PNBDCDXPQZPIPK
|
7.3 | IC50 | 3 | — | |
JHFJTTIYEGPPOW
|
7.3 | IC50 | 3 | — | |
RZJSWJLAOYUVRB
|
7.3 | IC50 | 3 | — | |
GVDYJBFFYVHNPA
|
7.3 | IC50 | 3 | — | |
XLHSLEFSSSWIGF
|
7.3 | IC50 | 3 | — | |
CXUFYCPSBOYQMV
|
7.3 | IC50 | 5 | — | |
YTTJKXSDNVYCBE
|
7.2 | IC50 | 3 | — | |
KGLWFPORHQPXJI
|
7.2 | IC50 | 3 | — | |
OTWGEGUQDHMDBA
|
7.2 | IC50 | 3 | — | |
RGKPUWYSUXLERI
|
7.2 | IC50 | 3 | — | |
QBINFJIYMSCWHV
|
7.2 | IC50 | 3 | — | |
YRYOEVHVROHLKR
|
7.2 | IC50 | 3 | — | |
DKEXUOIKEUTIAL
|
7.1 | IC50 | 3 | — | |
BERSUAQTWMUYMU
|
7.0 | IC50 | 3 | — | |
OYZYYVWBGXJDCM
|
7.0 | IC50 | 3 | — | |
XNLZFVQIZBXQNM
|
7.0 | IC50 | 3 | — | |
GHQHPTZESKRASB
|
7.0 | IC50 | 3 | — | |
JSONRPFPVGYCOB
|
6.9 | IC50 | 3 | — | |
HGAJCAYHMBFUDT
|
6.9 | IC50 | 3 | — | |
YJRWKOLRMSYZHE
|
6.9 | IC50 | 3 | — | |
QFGDRGRJMYSRIW
|
6.9 | IC50 | 3 | — | |
VPLRUYIVHZQYCE
|
6.9 | IC50 | 3 | — | |
RYTHFKJTOHUIJB
|
6.9 | IC50 | 3 | — | |
QAWHVZMZNTYGPK
|
6.8 | IC50 | 3 | — | |
QKWPGKWGXYCSIM
|
6.8 | IC50 | 3 | — | |
XFIGCAVKRPQHIW
|
6.8 | IC50 | 2 | — | |
CSXKZYFDPBVVPL
|
6.8 | IC50 | 2 | — | |
LMVAHLFZGWUGNF
|
6.7 | IC50 | 8 | Yes | |
MCKMGYSAHQYEDC
|
6.7 | IC50 | 3 | — | |
TYGCWIRHRMMCNF
|
6.7 | IC50 | 3 | — | |
HMRUGEAVJFRORJ
|
6.6 | IC50 | 3 | — | |
TYDGXGDYKRIRIF
|
6.5 | IC50 | 3 | — | |
PFDOYRBDNTWQJP
|
6.5 | IC50 | 2 | — | |
QVMWSFYCPYOKBR
|
6.5 | IC50 | 3 | — | |
LCQAIZAFSOZWRC
|
6.4 | IC50 | 8 | Yes | |
SZRCRQLPOHAVJL
|
6.3 | IC50 | 3 | — | |
TZDJIUGMUUUAQD
|
6.3 | IC50 | 3 | — | |
IXORERCONFMYQK
|
6.2 | IC50 | 3 | — | |
DJAZYXTUKHPMNT
|
6.2 | IC50 | 3 | — | |
XMTAJCWZZMFYID
|
6.1 | IC50 | 3 | — | |
ZGFXAJBFDCMHTM
|
6.0 | IC50 | 3 | Yes |