Target Details
| UniProt AC | Q8IYT8 |
|---|---|
| Gene Symbol | ULK2 |
| Protein Name | Serine/threonine-protein kinase ULK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12063 (ATG1-like_MIT1) PF21127 (ATG1-like_MIT2) PF00069 (Pkinase) |
Summary
- Multi-target molecules 45
- Clinical molecules 7
- Avg pChEMBL 7.09
KEGG Pathways (8)
Active Molecules (45)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KKISLZKMBSCLSS
|
9.0 | IC50 | 2 | — | |
UEZRAYLQPKCVRW
|
9.0 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
8.7 | Kd | 231 | Yes | |
KYPQUQARPVLCEI
|
8.6 | IC50 | 2 | — | |
QFSIUHFQOJVPBQ
|
8.6 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
YPJRHEKCFKOVRT
|
8.3 | Kd | 12 | — | |
DLCOOKRUECVLCI
|
7.9 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
7.9 | Kd | 201 | Yes | |
NHHQJBCNYHBUSI
|
7.7 | Kd | 220 | — | |
GVNUZZFMGGXPMN
|
7.5 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.5 | Kd | 200 | — | |
PFZRXJIYAFANHP
|
7.5 | IC50 | 4 | — | |
FIVNKJOGCQTGHE
|
7.4 | IC50 | 2 | — | |
LMPCYUMUDIOPBH
|
7.4 | IC50 | 2 | — | |
MGCUCAILCSYREM
|
7.4 | IC50 | 2 | — | |
UKBGBACORPRCGG
|
7.4 | IC50 | 17 | — | |
YRDHKIFCGOZTGD
|
7.4 | IC50 | 21 | — | |
PIQCTGMSNWUMAF
|
7.3 | Kd | 137 | Yes | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
OSVUGUHRKMMBSE
|
7.2 | Kd | 170 | — | |
CTNPALGJUAXMMC
|
7.2 | Kd | 151 | — | |
JOOXLOJCABQBSG
|
7.1 | Kd | 139 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
HFNKQEVNSGCOJV
|
6.7 | Kd | 65 | — | |
AQFMGFCVDBEMQE
|
6.7 | IC50 | 3 | — | |
VAVXGGRQQJZYBL
|
6.5 | IC50 | 8 | — | |
WVXNSAVVKYZVOE
|
6.5 | IC50 | 92 | — | |
ILNHHNVWAGBGGW
|
6.5 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
ZYLHCSSOEGIFAO
|
6.4 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
GUBJNPWVIUFSTR
|
6.3 | Kd | 103 | — | |
UBPYILGKFZZVDX
|
6.3 | Kd | 130 | Yes | |
BIIVYFLTOXDAOV
|
6.3 | Kd | 82 | Yes | |
BQROJYIEHOOQBY
|
6.3 | IC50 | 2 | — | |
YSCYSYZEYWGLFD
|
6.2 | IC50 | 2 | — | |
GWRHBTXTQFLVSP
|
6.2 | IC50 | 2 | — | |
NEXGBSJERNQRSV
|
6.2 | IC50 | 3 | — | |
HTSMUTPVZNMYSW
|
6.1 | IC50 | 2 | — | |
IGTBKTSITITXQX
|
6.1 | IC50 | 2 | — | |
JJEFZXFMIWYUFB
|
6.1 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |