Target Details
| UniProt AC | Q8IWQ3 |
|---|---|
| Gene Symbol | BRSK2 |
| Protein Name | Serine/threonine-protein kinase BRSK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21122 (KA1_BRSK) PF00069 (Pkinase) PF21115 (UBA_BRSK) |
Summary
- Multi-target molecules 16
- Clinical molecules 6
- Avg pChEMBL 7.19
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.5 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.5 | Kd | 213 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
MTLRBJOPNITTML
|
7.5 | Ki | 3 | — | |
NYUWMYQXNKUCSV
|
7.5 | Ki | 3 | — | |
ORDFJBYOBIZZSP
|
7.5 | Ki | 3 | — | |
MFAQYJIYDMLAIM
|
7.4 | Kd | 130 | Yes | |
CMWRPDHVGMHLSZ
|
7.0 | IC50 | 22 | — | |
GLDSKRNGVVYJAB
|
7.0 | Kd | 16 | — | |
SGZZQKMOFHIDKW
|
7.0 | Kd | 13 | — | |
LOGJQOUIVKBFGH
|
7.0 | IC50 | 11 | Yes | |
AILRADAXUVEEIR
|
6.9 | IC50 | 75 | — | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
YVVAPRJVYSYPJY
|
6.3 | Ki | 3 | — | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 91 | Yes |