Target Details
| UniProt AC | Q8IW41 |
|---|---|
| Gene Symbol | MAPKAPK5 |
| Protein Name | MAP kinase-activated protein kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 61
- Clinical molecules 6
- Avg pChEMBL 7.04
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (61)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HATNHAMXMKJCEI
|
6.1 | Ki | 9 | — | |
NLUPJKQOKWBWFC
|
6.1 | Ki | 69 | — | |
PZFVPUHGGQMWGD
|
6.1 | IC50 | 3 | — | |
SRUYMJRFVGLQDV
|
6.1 | Ki | 37 | — | |
UIARLYUEJFELEN
|
6.0 | Kd | 289 | Yes | |
DJUSDFVEBBYFFL
|
6.0 | Ki | 27 | — | |
DKSNLQYRZJKYOC
|
6.0 | Ki | 51 | — | |
FBWWNLBZZFVRQY
|
6.0 | Ki | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |