Target Details
| UniProt AC | Q8IW41 |
|---|---|
| Gene Symbol | MAPKAPK5 |
| Protein Name | MAP kinase-activated protein kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 61
- Clinical molecules 6
- Avg pChEMBL 7.04
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (61)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GIEOFRPQGSGOLC
|
9.5 | IC50 | 2 | — | |
HLFUJFUWDSXIPK
|
9.2 | IC50 | 2 | — | |
VFESYYJORSLMBC
|
9.0 | IC50 | 2 | — | |
SZMOXKFQHCNMQZ
|
8.9 | IC50 | 2 | — | |
JMCCHRFGZMNODA
|
8.8 | IC50 | 2 | — | |
VWNROJWIQIWFSP
|
8.8 | IC50 | 2 | — | |
LYZZMBVBMJMPFE
|
8.5 | IC50 | 2 | — | |
XWXSNJQHZKOICN
|
8.4 | IC50 | 2 | — | |
CMWRPDHVGMHLSZ
|
8.3 | IC50 | 22 | — | |
MFPICHSQTLJIFK
|
8.3 | IC50 | 2 | — | |
JMCCHRFGZMNODA
|
8.2 | IC50 | 2 | — | |
SBRNUAKQBCFNDP
|
8.2 | IC50 | 2 | — | |
HHFBDROWDBDFBR
|
8.1 | Kd | 40 | Yes | |
FEAAGBKEHOIVOC
|
8.0 | IC50 | 2 | — | |
MIKAKZKNMYZLDX
|
8.0 | Ki | 42 | — | |
CJLVRCRBVMSXBQ
|
7.7 | IC50 | 2 | — | |
ZJFVUVKJGZKTKC
|
7.7 | IC50 | 2 | — | |
AWZFCQRICMFIES
|
7.6 | IC50 | 9 | Yes | |
PGQVIPWLMNSOCQ
|
7.6 | IC50 | 2 | — | |
RLAJOHAIIACFAM
|
7.5 | IC50 | 13 | Yes | |
MWKSRKSEWLRPBL
|
7.4 | Kd | 1075 | — | |
JSKUWFIZUALZLX
|
7.2 | Ki | 33 | — | |
RJZDECGDCKOHBV
|
7.2 | Ki | 70 | — | |
HSKVRPZJBMXFDX
|
7.1 | Ki | 20 | — | |
OWFLADWRSCINST
|
7.1 | IC50 | 30 | — | |
JCFJQIHDZHHMQT
|
6.9 | Ki | 42 | — | |
NNQMSHWOTYMSDC
|
6.8 | IC50 | 3 | — | |
LRZYYIZFBXFSJB
|
6.7 | Ki | 69 | — | |
XJJYJNMNYDNXNO
|
6.7 | IC50 | 23 | — | |
FPQHXFMYXQZPSV
|
6.6 | Ki | 23 | — | |
GFOMFROIIBQABZ
|
6.6 | Ki | 7 | — | |
DKZYXHCYPUVGAF
|
6.6 | Kd | 112 | — | |
HKSZLNNOFSGOKW
|
6.6 | IC50 | 408 | — | |
XIOOJUQFJYPVLA
|
6.5 | Ki | 17 | — | |
CHYJUWDXSCFHON
|
6.5 | IC50 | 2 | — | |
BNLPAUPVSCPTDM
|
6.4 | Ki | 15 | — | |
GCYXEGSPUDSZJY
|
6.4 | Ki | 82 | — | |
LKUJDAHYLPICSE
|
6.4 | Ki | 24 | — | |
OLVBAUVSICCWEJ
|
6.4 | Ki | 39 | — | |
OWDRQHVEJIYVOI
|
6.4 | Ki | 47 | — | |
DKXHSOUZPMHNIZ
|
6.3 | IC50 | 51 | Yes | |
LOLPPWBBNUVNQZ
|
6.2 | Kd | 97 | Yes | |
BPJQSSSZFGZEOF
|
6.2 | Ki | 4 | — | |
IJNGXROUMFEKDB
|
6.2 | Ki | 39 | — | |
NFMGZVPRGVERNN
|
6.2 | Ki | 44 | — | |
PBNKREGCQAYWMQ
|
6.2 | Ki | 5 | — | |
STISJUSFFZAZMP
|
6.2 | Ki | 7 | — | |
ZQVQTUFEKLITNT
|
6.2 | Ki | 10 | — | |
QXPNJMHRUZCEAP
|
6.2 | IC50 | 14 | — | |
FUMCKNCUEAQHCV
|
6.1 | Ki | 103 | — |