Target Details
| UniProt AC | Q8IVW4 |
|---|---|
| Gene Symbol | CDKL3 |
| Protein Name | Cyclin-dependent kinase-like 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 7
- Clinical molecules 3
- Avg pChEMBL 7.1
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHQYAWLKOUOTQO
|
9.3 | IC50 | 20 | — | |
ODPGGGTTYSGTGO
|
8.3 | IC50 | 153 | — | |
ASGMFNBUXDJWJJ
|
6.8 | IC50 | 8 | — | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
UIARLYUEJFELEN
|
6.4 | Kd | 289 | Yes | |
MLDQJTXFUGDVEO
|
6.3 | Kd | 85 | Yes | |
ZECOHPFWGOCWLO
|
6.2 | IC50 | 5 | — |