Target Details
| UniProt AC | Q8IVH8 |
|---|---|
| Gene Symbol | MAP4K3 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 148
- Clinical molecules 18
- Avg pChEMBL 7.33
KEGG Pathways (1)
Active Molecules (148)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVYSKMXHCGBBQU
|
6.9 | IC50 | 2 | — | |
NSSDJHYKLWNDFG
|
6.9 | IC50 | 2 | — | |
LRINILBKXCVIMV
|
6.8 | IC50 | 3 | — | |
RVSSNRBUPQUIEG
|
6.8 | IC50 | 5 | — | |
OJPUQYTXGKTLEG
|
6.8 | IC50 | 2 | — | |
NGGXDEMZRGKNHG
|
6.8 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.8 | Kd | 191 | — | |
HGNARJFKBILTIL
|
6.8 | IC50 | 2 | — | |
SYMONOSPGXDMMP
|
6.8 | IC50 | 2 | — | |
WVUNYSQLFKLYNI
|
6.8 | Kd | 46 | Yes | |
HSEDUERTEYTVOT
|
6.8 | IC50 | 2 | — | |
KQCSODUJRAFWMC
|
6.8 | IC50 | 2 | — | |
YLGMPWWMPCGYBF
|
6.8 | IC50 | 2 | — | |
UZPJPJXENPGVRI
|
6.8 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
APVWQLVROLDAPP
|
6.7 | IC50 | 2 | — | |
DZIXRHJRLCGYPK
|
6.7 | IC50 | 3 | — | |
HZYIMGKDYXEJDM
|
6.7 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
GUBJNPWVIUFSTR
|
6.7 | Kd | 103 | — | |
AIKGYQDFIJRQIY
|
6.6 | IC50 | 9 | — | |
GIRPCUVQSUVBEK
|
6.6 | IC50 | 3 | — | |
OXIQDNRCSPETQV
|
6.6 | IC50 | 2 | — | |
OXIQDNRCSPETQV
|
6.6 | IC50 | 2 | — | |
NDXRAKYQSXBMOI
|
6.6 | IC50 | 2 | — | |
FTBMREIZHCLTPN
|
6.5 | IC50 | 3 | — | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
XZXHXSATPCNXJR
|
6.5 | Kd | 165 | Yes | |
UQBOLKBTUZZWBP
|
6.5 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
6.4 | Kd | 50 | — | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes | |
DYNHJHQFHQTFTP
|
6.4 | Kd | 38 | — | |
UJLAWZDWDVHWOW
|
6.3 | Kd | 4 | — | |
CYJPFBCHYRZAJL
|
6.3 | IC50 | 3 | — | |
OYONTEXKYJZFHA
|
6.3 | Kd | 69 | Yes | |
ALKJNCZNEOTEMP
|
6.3 | Kd | 55 | — | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
WGUVBZYIVFUKTF
|
6.2 | IC50 | 2 | — | |
APVWQLVROLDAPP
|
6.2 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
6.2 | Kd | 102 | Yes | |
KTEIFNKAUNYNJU
|
6.2 | IC50 | 6 | Yes | |
PBCZSGKMGDDXIJ
|
6.2 | Kd | 68 | Yes | |
RYYNGWLOYLRZLK
|
6.1 | Kd | 45 | — | |
KDKUVYLMPJIGKA
|
6.1 | Kd | 91 | Yes | |
ROEUNIAWGRPMCW
|
6.1 | IC50 | 2 | — | |
VXBAJLGYBMTJCY
|
6.1 | Kd | 34 | Yes | |
YKDKRNUADNJEHQ
|
6.0 | IC50 | 2 | — |