Target Details
| UniProt AC | Q8IVH8 |
|---|---|
| Gene Symbol | MAP4K3 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 148
- Clinical molecules 18
- Avg pChEMBL 7.33
KEGG Pathways (1)
Active Molecules (148)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYIQUCVGSYXGDF
|
7.7 | IC50 | 2 | — | |
BLXAELRPPPAZNL
|
7.7 | IC50 | 2 | — | |
OZYSZPHJVXITET
|
7.7 | IC50 | 2 | — | |
NCRZBWYKAOJRIJ
|
7.7 | IC50 | 2 | — | |
RPZBWDOAZIJTBM
|
7.7 | IC50 | 2 | — | |
JNCFZEVZRYWROV
|
7.7 | IC50 | 3 | — | |
IBOUTLNFGGJROR
|
7.6 | IC50 | 2 | — | |
WMOZCZVWHZOVFI
|
7.6 | IC50 | 2 | — | |
XHCPCYVQXFHJAU
|
7.6 | IC50 | 12 | — | |
NNJCLAJJCAILRT
|
7.6 | IC50 | 2 | — | |
CXIGTMXVRAHGKF
|
7.6 | IC50 | 2 | — | |
LMMPYMLTMDFZRW
|
7.5 | IC50 | 2 | — | |
OIJOOTMJWCNRQR
|
7.5 | IC50 | 2 | — | |
SXGLKAJWKHWEPI
|
7.5 | IC50 | 3 | — | |
XZVCLGAJVSWPFQ
|
7.5 | IC50 | 2 | — | |
PPGUULSJUXLSJS
|
7.4 | IC50 | 2 | — | |
RFUAALIUPJPJCJ
|
7.4 | IC50 | 2 | — | |
AIFRAZQXNNPZBV
|
7.4 | IC50 | 2 | — | |
VQYASORGHMGXQV
|
7.4 | IC50 | 2 | — | |
YPUUKVINJSRXQN
|
7.4 | IC50 | 2 | — | |
NHLRQGPSAURBBL
|
7.3 | IC50 | 3 | — | |
VRQMAABPASPXMW
|
7.3 | Kd | 10 | — | |
QAJMXNDGDLWDAN
|
7.3 | IC50 | 3 | — | |
AOJDKUXYLYKLKG
|
7.3 | IC50 | 2 | — | |
RWTXXGPUNDKBLW
|
7.2 | IC50 | 4 | — | |
QQWUGDVOUVUTOY
|
7.2 | Kd | 231 | Yes | |
OEOIPLGKLNBGHY
|
7.2 | IC50 | 2 | — | |
RMYZEICXBRZXFD
|
7.2 | IC50 | 2 | — | |
NRNCXXANURQNKO
|
7.1 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
7.1 | Kd | 114 | — | |
BRNMCVNQMQLRHM
|
7.1 | IC50 | 3 | — | |
KGMSWMZCIQWBHX
|
7.1 | IC50 | 3 | — | |
DSSNAGYVGTYAGH
|
7.1 | IC50 | 10 | — | |
NGGXDEMZRGKNHG
|
7.1 | IC50 | 2 | — | |
DTHDBWPUQXSBEE
|
7.1 | IC50 | 3 | — | |
YAPIPGOLZSTISM
|
7.0 | IC50 | 3 | — | |
KCVUUZPGZKJPAG
|
7.0 | IC50 | 2 | — | |
NSSDJHYKLWNDFG
|
7.0 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
7.0 | IC50 | 47 | — | |
CXQHYVUVSFXTMY
|
7.0 | Kd | 154 | — | |
IWFMUUASEIUTAN
|
7.0 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
7.0 | Kd | 149 | — | |
UIARLYUEJFELEN
|
7.0 | Kd | 289 | Yes | |
IPBBLOJPAZIORI
|
7.0 | IC50 | 2 | — | |
HGNARJFKBILTIL
|
6.9 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 91 | Yes | |
KQCSODUJRAFWMC
|
6.9 | IC50 | 2 | — | |
NIJYDRGSAYMLLQ
|
6.9 | IC50 | 2 | — | |
JBGWDRMZKMTPOT
|
6.9 | IC50 | 3 | — |