Target Details
| UniProt AC | Q8IVH8 |
|---|---|
| Gene Symbol | MAP4K3 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 148
- Clinical molecules 18
- Avg pChEMBL 7.33
KEGG Pathways (1)
Active Molecules (148)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.9 | IC50 | 408 | — | |
RVFYCRCCTDEQQD
|
9.3 | IC50 | 4 | — | |
LQUUWQNDKXYUCK
|
9.3 | IC50 | 2 | — | |
UUVGYKHBHXIMIM
|
9.1 | IC50 | 2 | — | |
XSIMOSPDULMWPL
|
8.8 | IC50 | 3 | — | |
VCCYOHCOICDUFL
|
8.5 | IC50 | 2 | — | |
DPLYERNYYUCIOC
|
8.4 | IC50 | 2 | — | |
REAMBIDJUBDLKK
|
8.4 | IC50 | 2 | — | |
IVKWJLVMIVBKDX
|
8.3 | IC50 | 2 | — | |
IVKWJLVMIVBKDX
|
8.3 | IC50 | 2 | — | |
SRTJPDZXTXFJPF
|
8.3 | IC50 | 2 | — | |
SVOVJJIXKQRGRV
|
8.3 | IC50 | 2 | — | |
ZTQCJUDBNICJBQ
|
8.3 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
8.3 | Kd | 130 | Yes | |
KHDZTOGFCVNLOZ
|
8.2 | IC50 | 2 | — | |
KHDZTOGFCVNLOZ
|
8.2 | IC50 | 2 | — | |
ZTSQSKNFQOTFNW
|
8.2 | IC50 | 2 | — | |
FYCAQERUJJTTFG
|
8.2 | IC50 | 2 | — | |
GFEVOBQWEKTOLR
|
8.2 | IC50 | 2 | — | |
JYDWXFPHARBUAB
|
8.2 | IC50 | 2 | — | |
OONFVLYMZFAOSH
|
8.2 | IC50 | 2 | — | |
ZZNHNGWYLUNNCT
|
8.1 | IC50 | 3 | — | |
JWNPDZNEKVCWMY
|
8.1 | Kd | 57 | Yes | |
SRHZWIQYIDTHNP
|
8.1 | IC50 | 2 | — | |
TWTKQXHGZXXULH
|
8.1 | IC50 | 2 | — | |
YGBJJONQEBBXHB
|
8.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.1 | Kd | 213 | — | |
MPFMLTBUDZGFRW
|
8.0 | IC50 | 2 | — | |
OIJOOTMJWCNRQR
|
8.0 | IC50 | 2 | — | |
WTTUTRXPNFTTPC
|
8.0 | IC50 | 3 | — | |
DETGKAHYPYOYLU
|
8.0 | IC50 | 2 | — | |
VPJYHGDUYQHMII
|
8.0 | IC50 | 2 | — | |
DKJPYCPAVXDNLO
|
7.9 | IC50 | 2 | — | |
OHVZGZMTULBSNX
|
7.9 | IC50 | 2 | — | |
VLNGPEMYJFURLB
|
7.9 | IC50 | 2 | — | |
WWENZKQHNDQUOA
|
7.9 | IC50 | 2 | — | |
FRGYOMQWHFXVEU
|
7.8 | IC50 | 3 | — | |
NNJCLAJJCAILRT
|
7.8 | IC50 | 2 | — | |
OZYSZPHJVXITET
|
7.8 | IC50 | 2 | — | |
ZUJPITIYCZFUQQ
|
7.8 | IC50 | 3 | — | |
QQVWHLARMCUHGI
|
7.8 | IC50 | 2 | — | |
FAYFPKOZAHXDIT
|
7.8 | IC50 | 2 | — | |
FTMLQXAVSYTOLC
|
7.8 | IC50 | 2 | — | |
MPFMLTBUDZGFRW
|
7.8 | IC50 | 2 | — | |
OSETUFDXSRDZOI
|
7.8 | IC50 | 2 | — | |
TTWHYLBRQRYBLK
|
7.8 | IC50 | 2 | — | |
BQRDIEUIHZRWEL
|
7.8 | IC50 | 2 | — | |
BTULSRXNMQZJDX
|
7.8 | IC50 | 2 | — | |
UNJMDMUQCPCLFE
|
7.8 | IC50 | 2 | — | |
VIXCHKGYFCCMEH
|
7.8 | IC50 | 2 | — |