Target Details
| UniProt AC | Q8IU80 |
|---|---|
| Gene Symbol | TMPRSS6 |
| Protein Name | Transmembrane protease serine 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00057 (Ldl_recept_a) PF01390 (SEA) PF00089 (Trypsin) |
Summary
- Multi-target molecules 77
- Clinical molecules 0
- Avg pChEMBL 8.01
Associated Diseases (1)
Active Molecules (77)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WHTKMCKEGVQWOA
|
7.9 | Ki | 2 | — | |
CWONXXSKOMNCJK
|
7.9 | Ki | 2 | — | |
NTPXWWJBHRPNJK
|
7.8 | Ki | 2 | — | |
YIQJMJSYXAKORA
|
7.7 | Ki | 2 | — | |
WUVZRGBAJWADEI
|
7.6 | Ki | 2 | — | |
DXBXFMGUSXIICV
|
7.5 | Ki | 2 | — | |
KYNIQQFIMSQNOR
|
7.4 | IC50 | 3 | — | |
ANOXPFVQQFERLB
|
7.3 | Ki | 2 | — | |
PUQNZQBNSIATMI
|
7.3 | Ki | 2 | — | |
WTBWSLUWVIEISS
|
7.2 | Ki | 2 | — | |
VBGVWKFAVGGQCH
|
7.1 | Ki | 4 | — | |
MHWPNEADOGSOHV
|
7.1 | Ki | 4 | — | |
ZLCINVZAICQINL
|
7.0 | Ki | 4 | — | |
QKFCYPKTTJCUSZ
|
6.8 | Ki | 8 | — | |
HJGBKSHYCKEJGU
|
6.8 | Ki | 4 | — | |
UXPIHWCOQPNKRS
|
6.7 | Ki | 3 | — | |
YLFDUDAILBTVGN
|
6.5 | Ki | 4 | — | |
BXXLERYKAMCOQH
|
6.5 | Ki | 3 | — | |
DJNNZKJZFCRFRX
|
6.4 | Ki | 4 | — | |
NRLHRRLCQPZVFI
|
6.4 | Ki | 3 | — | |
MKQBXZZBVTZVKV
|
6.3 | Ki | 2 | — | |
KWSMBEJYQLCPRA
|
6.3 | Ki | 6 | — | |
GJPPSRQGPWOXMV
|
6.2 | Ki | 3 | — | |
PBWYFIKBBSEVNZ
|
6.1 | Ki | 3 | — | |
XEYMSPYAMSNLLU
|
6.1 | Ki | 3 | — | |
VXUNFTCHIUPRIL
|
6.1 | Ki | 2 | — | |
VXMYQVUXZGHVKU
|
6.0 | Ki | 4 | — |