Target Details
| UniProt AC | Q8IM16 |
|---|---|
| Gene Symbol | PMIV |
| Protein Name | Plasmepsin IV |
| Organism | Plasmodium falciparum (isolate 3D7) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 72
- Clinical molecules 0
- Avg pChEMBL 7.21
Active Molecules (72)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NEZMJXSOLFCLPF
|
7.0 | IC50 | 3 | — | |
WPOCDUBRCAGMKZ
|
7.0 | IC50 | 5 | — | |
XDHIEWBZJYZMBU
|
7.0 | IC50 | 5 | — | |
LVPSHGRBVZDDGH
|
6.9 | IC50 | 2 | — | |
OBJZAQZWSSSART
|
6.9 | IC50 | 2 | — | |
XORQURWQFSWNRT
|
6.8 | IC50 | 2 | — | |
SNEOTYPQBVLWFB
|
6.8 | IC50 | 4 | — | |
KMZTVKCJBGRXHN
|
6.8 | IC50 | 3 | — | |
QJNWMBPHFFQJHB
|
6.7 | IC50 | 3 | — | |
RBRORTMADKIWQG
|
6.7 | IC50 | 2 | — | |
AZASRRIQYBSWGO
|
6.7 | IC50 | 3 | — | |
DVZXNZIZLMLECD
|
6.7 | IC50 | 3 | — | |
FTVBVWNZKYPGOY
|
6.7 | IC50 | 2 | — | |
SXLRRSVMGDBJCS
|
6.6 | IC50 | 4 | — | |
FXMLQRDALQEISW
|
6.4 | IC50 | 2 | — | |
GBIFQWZWWHMHND
|
6.3 | Ki | 2 | — | |
IBSOPQYKTQLOPF
|
6.3 | IC50 | 4 | — | |
WHGNYYBBVBYAKI
|
6.3 | IC50 | 2 | — | |
LBDNOWPWPVBZSU
|
6.3 | IC50 | 4 | — | |
FSMNBGWEFVUIAV
|
6.2 | IC50 | 4 | — | |
JVFLHYQEGOVVJW
|
6.1 | Ki | 2 | — | |
VEWFKNUERSAOIS
|
6.0 | IC50 | 3 | — |