Target Details
| UniProt AC | Q8IM16 |
|---|---|
| Gene Symbol | PMIV |
| Protein Name | Plasmepsin IV |
| Organism | Plasmodium falciparum (isolate 3D7) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 72
- Clinical molecules 0
- Avg pChEMBL 7.21
Active Molecules (72)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FAXGPCHRFPCXOO
|
9.5 | IC50 | 14 | — | |
IJSKTUPILCNGRO
|
8.2 | IC50 | 3 | — | |
MZZICJGCOVKCKO
|
8.1 | IC50 | 3 | — | |
QOGWENXQKQHNGY
|
8.0 | IC50 | 5 | — | |
SVHZZNJAPQRERT
|
8.0 | IC50 | 2 | — | |
SFYSZVJXKDRKMX
|
8.0 | IC50 | 4 | — | |
KXZKVZPYBMCFET
|
7.8 | IC50 | 5 | — | |
KKTYZYHUPKXLPL
|
7.8 | IC50 | 4 | — | |
KTBBODWOBFLAOA
|
7.8 | IC50 | 3 | — | |
QFSACLHXUZDWGE
|
7.8 | IC50 | 4 | — | |
PYBIHWRQNXYDCA
|
7.8 | IC50 | 3 | — | |
BQFXWLYPYJMHKI
|
7.7 | IC50 | 5 | — | |
JQYYZEGXJPYRRZ
|
7.7 | IC50 | 4 | — | |
WDONZLDRIZQKQI
|
7.6 | IC50 | 3 | — | |
HVMZYPNIRCCZDE
|
7.6 | IC50 | 3 | — | |
NKSLZHUZXVIXOR
|
7.6 | IC50 | 4 | — | |
WDKZPITZRFMOHK
|
7.6 | IC50 | 3 | — | |
JPXZSPXKQLJMSO
|
7.5 | IC50 | 4 | — | |
MYJBZTCPVQPNGD
|
7.5 | IC50 | 4 | — | |
BBOMNCJNDYMIAI
|
7.5 | IC50 | 3 | — | |
YDZUHIZMRBWWKY
|
7.5 | IC50 | 3 | — | |
RMTQJSAOWJWUPX
|
7.5 | Ki | 2 | — | |
YQCGITGXXMOUON
|
7.4 | IC50 | 3 | — | |
YAXAZYXURMLPBG
|
7.4 | IC50 | 3 | — | |
IBEPMPMHRMTCKS
|
7.4 | IC50 | 3 | — | |
CFOCZHLGHZFLCC
|
7.4 | IC50 | 3 | — | |
SWNKPSNZXWVRRI
|
7.4 | IC50 | 4 | — | |
NVOLQOLIKBYGFU
|
7.3 | IC50 | 3 | — | |
PSNGTIQWNUJCAN
|
7.3 | IC50 | 6 | — | |
HUAHAYIWRIITDA
|
7.3 | IC50 | 2 | — | |
KGUVGCXOHCGRTK
|
7.3 | IC50 | 3 | — | |
LENHFBMFSSMDGV
|
7.3 | IC50 | 3 | — | |
MHNXYKUQICQQIS
|
7.2 | IC50 | 3 | — | |
NYVBCXDVWVZUQX
|
7.2 | IC50 | 4 | — | |
GBIXFQIQEIDDLN
|
7.2 | IC50 | 3 | — | |
KKROSRYNPGAQGH
|
7.2 | IC50 | 5 | — | |
YWKQULGMWFKKBB
|
7.2 | IC50 | 4 | — | |
FGOYNOLZZKCCHM
|
7.2 | IC50 | 4 | — | |
QRADGLCPTLHEAC
|
7.2 | IC50 | 3 | — | |
LZAOFFKQJKSBBG
|
7.2 | IC50 | 3 | — | |
GYISSNTWJQZCHG
|
7.1 | IC50 | 2 | — | |
GJKQZFJOCTXOHB
|
7.1 | IC50 | 2 | — | |
GBKSTUMREALLDP
|
7.1 | IC50 | 2 | — | |
CLPJFWBCLJHKBP
|
7.1 | IC50 | 3 | — | |
CPENPHULHCEEFK
|
7.0 | IC50 | 3 | — | |
ZHLPFTVHHADULF
|
7.0 | IC50 | 4 | — | |
DHCRLVYXJVDQLW
|
7.0 | IC50 | 2 | — | |
CFMJBMZVLYGUOI
|
7.0 | IC50 | 4 | — | |
IGDREXIRARRTCV
|
7.0 | IC50 | 2 | — | |
LOBCJUCVSNWELD
|
7.0 | IC50 | 3 | — |