Target Details
| UniProt AC | Q8IL11 |
|---|---|
| Gene Symbol | LAP |
| Protein Name | Leucine aminopeptidase |
| Organism | Plasmodium falciparum (isolate 3D7) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00883 (Peptidase_M17) |
Summary
- Multi-target molecules 18
- Clinical molecules 0
- Avg pChEMBL 9.46
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VLCYMYIBZFAFLM
|
11.1 | Ki | 2 | — | |
XHKYHEBAKPKAIX
|
11.0 | Ki | 2 | — | |
DZQODXUHSICRDF
|
10.9 | Ki | 2 | — | |
MDRSEUSHAKMGJK
|
10.8 | Ki | 2 | — | |
ZZJQASGOLBFQNU
|
10.8 | Ki | 2 | — | |
MYWRQDNAPJWUSO
|
10.7 | Ki | 2 | — | |
CUWFEJVIZZQNCM
|
10.6 | Ki | 2 | — | |
PGHJYUATTUXMSH
|
10.5 | Ki | 2 | — | |
OQNJTJVDXVRAAX
|
10.5 | Ki | 2 | — | |
BCTKXGZXZRVSQJ
|
10.4 | Ki | 2 | — | |
ZZLMORFDMAOBOY
|
10.3 | Ki | 2 | — | |
LGMNTGBSDLNSAJ
|
9.8 | Ki | 2 | — | |
STVSJGZHUJJREA
|
8.0 | Ki | 4 | — | |
QELOIXSGJMIHBZ
|
7.9 | Ki | 3 | — | |
QELOIXSGJMIHBZ
|
7.9 | Ki | 4 | — | |
OKPQYTOWYYKMHU
|
7.1 | Ki | 2 | — | |
FSULYXCULMDLOG
|
6.0 | IC50 | 2 | — | |
XGHUJWTXGMRXEL
|
6.0 | IC50 | 3 | — |