Target Details
| UniProt AC | Q8IIL0 |
|---|---|
| Gene Symbol | FP3 |
| Protein Name | Falcipain-3 |
| Organism | Plasmodium falciparum (isolate 3D7) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 22
- Clinical molecules 1
- Avg pChEMBL 6.64
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ASRBKZHDORPEHO
|
7.7 | IC50 | 5 | — | |
PNBVCCNBLDPOTA
|
7.2 | IC50 | 2 | — | |
IMTIJVSUXSYPRE
|
7.1 | IC50 | 2 | — | |
OLNJKAXRBXUBTB
|
7.0 | IC50 | 10 | Yes | |
QTDXHJIDZCYDHI
|
7.0 | IC50 | 2 | — | |
KGWCBORIZBPTEG
|
6.9 | IC50 | 4 | — | |
LTLYEAJONXGNFG
|
6.9 | IC50 | 9 | — | |
ZJLUYWUYIFDQKX
|
6.9 | IC50 | 2 | — | |
KMVGYYSPDSERNQ
|
6.9 | IC50 | 2 | — | |
VHDAHAMWVNXMSP
|
6.9 | IC50 | 4 | — | |
YHKOHOCWRAYTOU
|
6.6 | IC50 | 2 | — | |
LNGNOOFNSJGQRC
|
6.4 | IC50 | 2 | — | |
IEUSTTSJUZYCDI
|
6.3 | IC50 | 2 | — | |
MCXBQDQFTXLDCH
|
6.3 | IC50 | 2 | — | |
ONFPDHLEGKDYNI
|
6.3 | IC50 | 2 | — | |
VHDAHAMWVNXMSP
|
6.3 | IC50 | 7 | — | |
MAZZRZYOVBSDFO
|
6.3 | IC50 | 2 | — | |
PEOGBPZOQJURKT
|
6.3 | IC50 | 2 | — | |
ZQTRZEVHJUGKTF
|
6.3 | IC50 | 2 | — | |
DNVSLZJMWYZCRS
|
6.3 | IC50 | 2 | — | |
KYZFVJVVYWBTSG
|
6.1 | IC50 | 2 | — | |
ZQTRZEVHJUGKTF
|
6.0 | IC50 | 2 | — |