Target Details
| UniProt AC | Q8IAS0 |
|---|---|
| Gene Symbol | PMX |
| Protein Name | Plasmepsin X |
| Organism | Plasmodium falciparum (isolate 3D7) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 31
- Clinical molecules 0
- Avg pChEMBL 8.47
Active Molecules (31)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZSZSSSHEMYULPX
|
10.5 | IC50 | 2 | — | |
VRULKACKCWLXKD
|
10.2 | IC50 | 2 | — | |
DMZSBXNGCZIMPB
|
10.2 | IC50 | 2 | — | |
HRWUWCOIOZJWDO
|
9.5 | IC50 | 2 | — | |
MDTDXKZXNMWATA
|
9.4 | IC50 | 2 | — | |
PYBIHWRQNXYDCA
|
9.4 | IC50 | 3 | — | |
CTDJSVJRZFOZMC
|
9.2 | IC50 | 2 | — | |
IBEPMPMHRMTCKS
|
8.6 | IC50 | 3 | — | |
GYISSNTWJQZCHG
|
8.4 | IC50 | 2 | — | |
FGOYNOLZZKCCHM
|
8.4 | IC50 | 4 | — | |
GBKSTUMREALLDP
|
8.3 | IC50 | 2 | — | |
KMZTVKCJBGRXHN
|
8.3 | IC50 | 3 | — | |
QLAIIPJYEKWZKY
|
8.3 | IC50 | 2 | — | |
MHNXYKUQICQQIS
|
8.2 | IC50 | 3 | — | |
AZASRRIQYBSWGO
|
8.2 | IC50 | 3 | — | |
RBRORTMADKIWQG
|
8.2 | IC50 | 2 | — | |
AWSRDDSRQUJMAJ
|
8.2 | IC50 | 2 | — | |
NRQARCCHBBGTDO
|
8.2 | IC50 | 4 | — | |
GKMRULMLMQTRPR
|
8.1 | IC50 | 2 | — | |
QRADGLCPTLHEAC
|
8.1 | IC50 | 3 | — | |
ADUSWAORGLLWAE
|
8.1 | IC50 | 2 | — | |
RUZADINCVKIRSK
|
8.1 | IC50 | 2 | — | |
WYTXSWVPAXOIQI
|
8.0 | IC50 | 2 | — | |
NQNIOGFFUJELEC
|
8.0 | IC50 | 2 | — | |
ILMXPKBEEIKSAB
|
8.0 | IC50 | 2 | — | |
GIRFFPCRVUPHFZ
|
8.0 | IC50 | 2 | — | |
LBDNOWPWPVBZSU
|
8.0 | IC50 | 4 | — | |
UYHOZHWPCPSMFR
|
8.0 | IC50 | 2 | — | |
XPWMQRABBPYMQE
|
7.8 | IC50 | 2 | — | |
PGXFAIZJBZYGGS
|
7.6 | IC50 | 2 | — | |
RKULQZNRBARYRL
|
7.2 | IC50 | 2 | — |