Target Details
| UniProt AC | Q8I6Z5 |
|---|---|
| Gene Symbol | PMV |
| Protein Name | Plasmepsin V |
| Organism | Plasmodium falciparum (isolate 3D7) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00026 (Asp) PF14543 (TAXi_N) |
Summary
- Multi-target molecules 19
- Clinical molecules 14
- Avg pChEMBL 7.49
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VAHRPHLZONNTFF
|
9.4 | IC50 | 2 | — | |
DVJGXMUWYFGXAS
|
9.4 | pIC50 | 4 | Yes | |
AWOGCPXUTJBQEG
|
8.8 | pIC50 | 3 | Yes | |
PMFBLJXNSAHZSG
|
8.2 | pIC50 | 3 | Yes | |
NGBKFLTYGSREKK
|
8.1 | pIC50 | 6 | Yes | |
CSKGFHNQMOIAFM
|
8.0 | pIC50 | 4 | Yes | |
PQZHZCPKSLRZNY
|
7.7 | IC50 | 2 | — | |
ICRSIRKIELQUKD
|
7.6 | IC50 | 2 | — | |
BHGWRSHPZOLPAL
|
7.5 | IC50 | 2 | — | |
RXCRNUBYZRKEGC
|
7.5 | pIC50 | 3 | Yes | |
OLNJKAXRBXUBTB
|
7.1 | pIC50 | 10 | Yes | |
YYDQGTWJPADAKS
|
7.1 | pIC50 | 3 | Yes | |
JNRHNGGTJOBXHL
|
7.0 | pIC50 | 3 | Yes | |
WJFAAUIYJQVQJJ
|
7.0 | pIC50 | 3 | Yes | |
PGOQBJBMASKTEL
|
6.7 | pIC50 | 3 | Yes | |
QVDJMLQSYRSZKC
|
6.7 | pIC50 | 6 | Yes | |
YIRUASIRQWZPIZ
|
6.6 | pIC50 | 2 | Yes | |
PSNGTIQWNUJCAN
|
6.0 | IC50 | 6 | — | |
URUPDOIKTMCJNA
|
6.0 | pIC50 | 2 | Yes |