Target Details
| UniProt AC | Q86YV6 |
|---|---|
| Gene Symbol | MYLK4 |
| Protein Name | Myosin light chain kinase family member 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 43
- Clinical molecules 7
- Avg pChEMBL 6.76
KEGG Pathways (10)
Active Molecules (43)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VCZRYZZCLOMGOV
|
8.7 | IC50 | 4 | — | |
KAEJBHCXBMUJRI
|
8.2 | IC50 | 2 | — | |
VUQUBDXLGAPBGS
|
8.2 | IC50 | 2 | — | |
FAUVGWZEHNGPFI
|
7.9 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
7.8 | Kd | 201 | Yes | |
AHQYMFOEOWUTJB
|
7.8 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
CTNPALGJUAXMMC
|
7.5 | Kd | 151 | — | |
YZVSEVMXAIJHKO
|
7.4 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.3 | IC50 | 408 | — | |
RSJLKPAADCXPOZ
|
7.3 | IC50 | 2 | — | |
WNFAWYDESPZZIJ
|
7.3 | IC50 | 2 | — | |
XOCCIJUVHIYNCB
|
7.2 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
7.1 | Kd | 137 | Yes | |
IDNFFZUHFOQNRQ
|
7.1 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.9 | Kd | 139 | — | |
DORZPJWJOBMQKC
|
6.9 | IC50 | 9 | — | |
YYLKKYCXAOBSRM
|
6.8 | Kd | 191 | — | |
WNFAWYDESPZZIJ
|
6.8 | IC50 | 2 | — | |
AXRCEOKUDYDWLF
|
6.6 | Kd | 31 | — | |
XCOSAQGGGZDYJN
|
6.4 | Kd | 11 | — | |
ATWJOSDBVRWRHS
|
6.4 | IC50 | 5 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
HKSZLNNOFSGOKW
|
6.3 | Kd | 213 | — | |
ANGDJJFQAIUXQR
|
6.3 | IC50 | 2 | — | |
DYGYVRRCXQMZJC
|
6.3 | IC50 | 2 | — | |
LTXBFJFJUIJOQE
|
6.3 | IC50 | 3 | — | |
MMLWXRJMBOZWCU
|
6.3 | IC50 | 2 | — | |
NHCZWHGCNNIQHP
|
6.3 | IC50 | 2 | — | |
UDWJOFBRPYNJOD
|
6.3 | IC50 | 2 | — | |
WFKLCCZTEPHYPI
|
6.3 | IC50 | 2 | — | |
YKHAIGSLIKEHTC
|
6.3 | IC50 | 2 | — | |
ZFBYIIFQXUFBCC
|
6.3 | IC50 | 2 | — | |
NXWXUDHOUKWAQU
|
6.2 | Kd | 16 | — | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 91 | Yes | |
PSPFQEBFYXJZEV
|
6.2 | Kd | 10 | — | |
LHNIIDJUOCFXAP
|
6.1 | Kd | 20 | Yes | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |