Target Details
| UniProt AC | Q86Y07 |
|---|---|
| Gene Symbol | VRK2 |
| Protein Name | Serine/threonine-protein kinase VRK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 7
- Clinical molecules 2
- Avg pChEMBL 6.66
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTEKTGDVSARYDS
|
7.8 | Ki | 3 | — | |
DTEKTGDVSARYDS
|
7.5 | Ki | 11 | — | |
BIIVYFLTOXDAOV
|
7.2 | Kd | 82 | Yes | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |