Target Details
| UniProt AC | Q86X55 |
|---|---|
| Gene Symbol | CARM1 |
| Protein Name | Histone-arginine methyltransferase CARM1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11531 (CARM1) PF06325 (PrmA) PF22528 (PRMT_C) |
Summary
- Multi-target molecules 120
- Clinical molecules 0
- Avg pChEMBL 7.33
KEGG Pathways (1)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHEBNMWUAGLPPM
|
6.6 | IC50 | 2 | — | |
FUUQRIOHQLDOTR
|
6.6 | IC50 | 2 | — | |
AMPQIHZOWIDPQA
|
6.5 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.5 | Kd | 599 | — | |
GZLKEWKXXDOJMT
|
6.5 | IC50 | 2 | — | |
WTEPBGJODXCGET
|
6.5 | IC50 | 2 | — | |
ZDCXQYXHINCUOB
|
6.5 | IC50 | 2 | — | |
UXQWECXRONTUQW
|
6.5 | IC50 | 3 | — | |
QTNIFNOIKLRHGJ
|
6.4 | IC50 | 2 | — | |
UBOFQOGNZXZZPE
|
6.4 | IC50 | 2 | — | |
ZJUKTBDSGOFHSH
|
6.4 | Ki | 22 | — | |
KQGWUTGYBNKPKE
|
6.4 | IC50 | 2 | — | |
HVDMIAFOVVMNJF
|
6.3 | IC50 | 4 | — | |
NSMVLEXMOMOBHV
|
6.3 | IC50 | 2 | — | |
OEUKIVBCINJEJS
|
6.2 | IC50 | 2 | — | |
SVJIZDDQCMAIMW
|
6.2 | IC50 | 2 | — | |
DICKVPVLKDVBPQ
|
6.2 | IC50 | 3 | — | |
GJPQENHVEQGHGP
|
6.2 | Kd | 3 | — | |
OVCOWLKXRNBYMI
|
6.0 | IC50 | 2 | — | |
PCNDXYHWLSHXMV
|
6.0 | IC50 | 2 | — |