Target Details
| UniProt AC | Q86X55 |
|---|---|
| Gene Symbol | CARM1 |
| Protein Name | Histone-arginine methyltransferase CARM1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11531 (CARM1) PF06325 (PrmA) PF22528 (PRMT_C) |
Summary
- Multi-target molecules 120
- Clinical molecules 0
- Avg pChEMBL 7.33
KEGG Pathways (1)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HBOJWAYLSJLULG
|
7.5 | IC50 | 5 | — | |
KAVMHQFWHGHFMI
|
7.5 | IC50 | 2 | — | |
YDVOPOIVFHFPTA
|
7.5 | IC50 | 2 | — | |
MPASEZSHHLMDOX
|
7.4 | IC50 | 2 | — | |
MOPCOJLFDMFKCS
|
7.4 | IC50 | 2 | — | |
NSMVLEXMOMOBHV
|
7.4 | IC50 | 2 | — | |
HYQMJLIWAPDIFI
|
7.4 | IC50 | 2 | — | |
LPBWALAEOJUKMO
|
7.4 | IC50 | 2 | — | |
SVGZJNSANYCCJO
|
7.4 | IC50 | 2 | — | |
SYRKWCSTKUNNAO
|
7.4 | IC50 | 2 | — | |
RWVFEGDWAMZZBR
|
7.3 | IC50 | 2 | — | |
JMANMSSINYWBCS
|
7.3 | IC50 | 2 | — | |
ICLYSKVLWUOLLZ
|
7.3 | IC50 | 2 | — | |
KSSCHHFJLLWFFW
|
7.3 | IC50 | 2 | — | |
DUACCTUMSKZJAG
|
7.3 | IC50 | 2 | — | |
QVOKJKWHZRTVQQ
|
7.3 | IC50 | 3 | — | |
FPMCBNOZDJXPHM
|
7.3 | IC50 | 2 | — | |
IYQWSDAAFFNNME
|
7.3 | IC50 | 2 | — | |
FZVDFKGBRORXNX
|
7.2 | IC50 | 2 | — | |
MTWABGJHHGHDEQ
|
7.2 | IC50 | 2 | — | |
XCZUYGFLWBJNCB
|
7.2 | IC50 | 4 | — | |
QTNIFNOIKLRHGJ
|
7.2 | IC50 | 2 | — | |
XJTRJDJVJPHIJZ
|
7.2 | IC50 | 2 | — | |
YPDKIXXYOHVHBD
|
7.2 | IC50 | 3 | — | |
PKUZYKBLICNLDH
|
7.2 | IC50 | 2 | — | |
WPAHUPFRZFNUKC
|
7.1 | IC50 | 2 | — | |
VWJBIFGWCPEUEE
|
7.1 | IC50 | 2 | — | |
WFHFRZYKQWQVOL
|
7.1 | IC50 | 3 | — | |
LUBCTIQAZDQPJR
|
7.1 | IC50 | 5 | — | |
YWNMOMVIHTWXNN
|
7.1 | IC50 | 2 | — | |
HWAIOOIUDDHXSO
|
7.0 | IC50 | 2 | — | |
VYBORVUUKYMIGQ
|
7.0 | IC50 | 2 | — | |
WBYJDMKBPXSKDH
|
7.0 | IC50 | 2 | — | |
CGRVFRVDHNMDLY
|
7.0 | IC50 | 2 | — | |
FWIUJOSFDRYPNT
|
7.0 | IC50 | 2 | — | |
LQMZTSHUQPYZKP
|
7.0 | IC50 | 2 | — | |
VZZSAYLJCKTKMS
|
7.0 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.0 | Kd | 1075 | — | |
HDLMOUYGUDJTRP
|
6.9 | IC50 | 3 | — | |
ZHKZDMWVMUFTSS
|
6.9 | IC50 | 2 | — | |
JUDPMRRWNRXOOF
|
6.9 | IC50 | 2 | — | |
GJSRTOARMZMCJN
|
6.9 | IC50 | 2 | — | |
CBLOJJICRSGZRU
|
6.9 | IC50 | 4 | — | |
UDFJXRJYAZANFF
|
6.8 | IC50 | 3 | — | |
ZYQFUTZIWVTGCH
|
6.8 | IC50 | 2 | — | |
QGIYMANUGUDANL
|
6.8 | IC50 | 2 | — | |
CWSANINJEGUUDR
|
6.8 | IC50 | 2 | — | |
VZDPLMKEFMWBMM
|
6.8 | IC50 | 5 | — | |
YHJMIEBEURJANR
|
6.8 | IC50 | 2 | — | |
YVYXQOZXGQSVIU
|
6.7 | IC50 | 2 | — |