Target Details
| UniProt AC | Q86X55 |
|---|---|
| Gene Symbol | CARM1 |
| Protein Name | Histone-arginine methyltransferase CARM1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11531 (CARM1) PF06325 (PrmA) PF22528 (PRMT_C) |
Summary
- Multi-target molecules 120
- Clinical molecules 0
- Avg pChEMBL 7.33
KEGG Pathways (1)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UMKLFWMQTDMELK
|
8.7 | IC50 | 5 | — | |
CDHNSYFOBQQCHE
|
8.6 | IC50 | 2 | — | |
OQFRQLWUXSTHHK
|
8.6 | IC50 | 3 | — | |
PMLVTAUALHGTDV
|
8.6 | IC50 | 2 | — | |
QRIOWSCVJSHXMY
|
8.6 | IC50 | 2 | — | |
WYAODYBTCNOEPW
|
8.5 | IC50 | 2 | — | |
XJYXSHKKYORCSG
|
8.5 | IC50 | 2 | — | |
DVIUIRPCVXVFSX
|
8.4 | IC50 | 3 | — | |
RGVCBFLWXVBFNB
|
8.4 | IC50 | 2 | — | |
DVZZYZNFLHFCPI
|
8.3 | IC50 | 7 | — | |
WYAODYBTCNOEPW
|
8.3 | IC50 | 2 | — | |
CNMWTZSRTFSQJJ
|
8.2 | IC50 | 5 | — | |
KSPVNKWKRYGRDT
|
8.2 | IC50 | 2 | — | |
DYDJINHRKAERSQ
|
8.1 | IC50 | 2 | — | |
MOPCOJLFDMFKCS
|
8.1 | IC50 | 4 | — | |
ILHAASUEJBNZOF
|
8.0 | IC50 | 2 | — | |
PFNIKRLIXXKHOH
|
7.9 | IC50 | 2 | — | |
UMKLFWMQTDMELK
|
7.9 | IC50 | 2 | — | |
KUAIUYDMQDZPEQ
|
7.9 | IC50 | 2 | — | |
KOVXGJRGKPPNMB
|
7.8 | IC50 | 2 | — | |
DBWNSLHFKVEMFR
|
7.8 | IC50 | 2 | — | |
ILHAASUEJBNZOF
|
7.8 | IC50 | 2 | — | |
LAWOIDJHIVKWDO
|
7.8 | IC50 | 2 | — | |
SPEGERVLTUWZPA
|
7.8 | IC50 | 5 | — | |
JYIRWTZMMGLPFI
|
7.8 | IC50 | 2 | — | |
MJBSRPRJLFEYAZ
|
7.8 | IC50 | 2 | — | |
GBDIISBIAOHVMJ
|
7.8 | IC50 | 2 | — | |
HGLUYHIGDAHROE
|
7.8 | IC50 | 2 | — | |
QRXRBRDDXIISAI
|
7.8 | IC50 | 2 | — | |
SIOCLBFQLPHPJM
|
7.8 | IC50 | 2 | — | |
UOYQDRFGWGTDNI
|
7.8 | IC50 | 2 | — | |
MOWUZOHGLGUMND
|
7.8 | IC50 | 2 | — | |
ZKGHABBSYZLSAM
|
7.8 | IC50 | 2 | — | |
FOPJHWSUFHQCBW
|
7.7 | IC50 | 2 | — | |
VVGWNMSYHCMOPA
|
7.7 | IC50 | 2 | — | |
MBBYYSNFGWIUIY
|
7.7 | IC50 | 2 | — | |
HGLUYHIGDAHROE
|
7.7 | IC50 | 2 | — | |
DMXKZVDCWGJXLG
|
7.7 | IC50 | 2 | — | |
NHEFIVVNRQJHSA
|
7.7 | IC50 | 2 | — | |
FMTVWAGUJRUAKE
|
7.6 | IC50 | 5 | — | |
SXNQENMPTCVHFW
|
7.6 | IC50 | 2 | — | |
BFQFZLZUYSLBRQ
|
7.6 | IC50 | 2 | — | |
QBRANFNGHJILEL
|
7.6 | IC50 | 2 | — | |
QNBYZAPNKWTVTR
|
7.6 | IC50 | 2 | — | |
OLFLGFYCUQONAR
|
7.6 | IC50 | 3 | — | |
AAFISRHSQOGOSG
|
7.5 | IC50 | 2 | — | |
JXTSMPSQQKIELG
|
7.5 | IC50 | 2 | — | |
XSOARJRAIKUXSE
|
7.5 | IC50 | 2 | — | |
SPSRJAZORUFUOI
|
7.5 | IC50 | 2 | — | |
GMMYYQFKUWMMHS
|
7.5 | IC50 | 2 | — |