Target Details
| UniProt AC | Q86V86 |
|---|---|
| Gene Symbol | PIM3 |
| Protein Name | Serine/threonine-protein kinase pim-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,417
- Clinical molecules 10
- Avg pChEMBL 8.16
Active Molecules (1,417)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NESXNWQYGLDRMW
|
8.9 | IC50 | 3 | — | |
NLOZLPYLNHZXJD
|
8.9 | IC50 | 3 | — | |
SYPBNOXLIVCNCJ
|
8.9 | Ki | 3 | — | |
UORSWGPLCPBYOP
|
8.9 | IC50 | 3 | — | |
VJXUXTWQBIILQL
|
8.9 | Ki | 3 | — | |
LKVRXZVHFRHSKB
|
8.9 | IC50 | 3 | — | |
MYYHUGRZNUGCBD
|
8.9 | Ki | 3 | — | |
FTQIZXVNFDCIQI
|
8.8 | Ki | 3 | — | |
JLRFGUCJKRWAIB
|
8.8 | IC50 | 3 | — | |
SMWFSPOWWDSJEB
|
8.8 | IC50 | 3 | — | |
FKRJLOFLENGVAA
|
8.8 | IC50 | 3 | — | |
KEQAECANTREWKS
|
8.8 | IC50 | 3 | — | |
LLNGTXPGUYSOTJ
|
8.8 | IC50 | 3 | — | |
NIOMNUVZCQNZEN
|
8.8 | IC50 | 3 | — | |
ZBNXMASDPWDPMD
|
8.8 | IC50 | 3 | — | |
DXLJDEPUAKIDEU
|
8.8 | IC50 | 3 | — | |
KYXJMCQQNZDWIT
|
8.8 | IC50 | 3 | — | |
NLOZLPYLNHZXJD
|
8.8 | IC50 | 3 | — | |
OLKXVDKTEYJKPA
|
8.8 | IC50 | 3 | — | |
ROWCDUKNAFYOMJ
|
8.8 | IC50 | 3 | — | |
XTEHYWPWYQSFDO
|
8.8 | IC50 | 3 | — | |
MMQGQQIWWVVFQW
|
8.8 | IC50 | 3 | — | |
QMBLOFSJYILYLC
|
8.8 | IC50 | 3 | — | |
JBUOFUIXSMJURC
|
8.8 | IC50 | 3 | — | |
NWDVLGCDUFSSHA
|
8.8 | IC50 | 3 | — | |
UPNOOQUTVLYBIK
|
8.8 | Ki | 3 | — | |
AYUREZCMYVPMPV
|
8.8 | IC50 | 3 | — | |
ISRJLVCSRJCNHO
|
8.8 | Ki | 3 | — | |
JVMZLXCDQMDOEH
|
8.8 | IC50 | 3 | — | |
WAGFUTAXHIKUFA
|
8.8 | IC50 | 3 | — | |
AVWIQATUPWLNJO
|
8.8 | IC50 | 3 | — | |
GANOQVZZUSOYDP
|
8.8 | IC50 | 3 | — | |
MXLKCGYBUFWTAU
|
8.8 | IC50 | 3 | — | |
BNXXSPKXSUAPBT
|
8.8 | IC50 | 3 | — | |
FVOUGHZKLGXVGD
|
8.8 | IC50 | 3 | — | |
KRMOAWBSZVZSIA
|
8.8 | IC50 | 3 | — | |
ANEQDQCTWAKZMN
|
8.8 | Ki | 3 | — | |
DPERSSXJBGKIEL
|
8.8 | Ki | 3 | — | |
FLPSOVPOQWHOJV
|
8.8 | IC50 | 3 | — | |
YXBOQTUJWONSJX
|
8.8 | IC50 | 3 | — | |
GHJCZGQHMLEEKQ
|
8.7 | IC50 | 3 | — | |
JFRTUZNKHJJSEH
|
8.7 | Ki | 3 | — | |
KTWFLQDWXPMQKC
|
8.7 | IC50 | 3 | — | |
WUTCYYSJWLOLPF
|
8.7 | IC50 | 3 | — | |
XYDAVXLWFUQNSH
|
8.7 | IC50 | 7 | — | |
YKRVUDKGPNZLLY
|
8.7 | Ki | 3 | — | |
CKRMSGUCWWVREC
|
8.7 | IC50 | 3 | — | |
MCUJKPPARUPFJM
|
8.7 | IC50 | 3 | — | |
MCUJKPPARUPFJM
|
8.7 | IC50 | 11 | — | |
WYFWPBSKKJQUBK
|
8.7 | IC50 | 3 | — |