Target Details
| UniProt AC | Q86V86 |
|---|---|
| Gene Symbol | PIM3 |
| Protein Name | Serine/threonine-protein kinase pim-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,417
- Clinical molecules 10
- Avg pChEMBL 8.16
Active Molecules (1,417)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JYUCZTGADIKZPX
|
8.2 | IC50 | 3 | — | |
QYFGCYLEXSUIII
|
8.2 | IC50 | 3 | — | |
HTMBVCFZCSVVSW
|
8.2 | IC50 | 3 | — | |
ILVKLFOUGPBUMK
|
8.2 | IC50 | 3 | — | |
LWHTZTIHIFBTMB
|
8.2 | IC50 | 3 | — | |
QOBRNBJEEWVJLW
|
8.2 | IC50 | 3 | — | |
VBZISNIVQBAKDD
|
8.2 | Ki | 3 | — | |
PLLDESOQBJZGSQ
|
8.2 | IC50 | 3 | — | |
AXPHZYUNEZZRPW
|
8.2 | IC50 | 3 | — | |
BGYKECRMNHZETP
|
8.2 | IC50 | 3 | — | |
CGBJYLPDYMUGJF
|
8.2 | IC50 | 3 | — | |
FRVOCFJDZQHLPC
|
8.2 | IC50 | 3 | — | |
GMLWQFRZINHDEH
|
8.2 | IC50 | 3 | — | |
GQCHSJRNLCGUAC
|
8.2 | IC50 | 3 | — | |
GTHLJKKDZJPZLZ
|
8.2 | IC50 | 3 | — | |
HJJCPVZAEJNRGD
|
8.2 | IC50 | 3 | — | |
HQWHAKOOAUIEHY
|
8.2 | IC50 | 3 | — | |
JTESMRSKGHICMR
|
8.2 | IC50 | 3 | — | |
JXHFSTVXTDOYNC
|
8.2 | IC50 | 3 | — | |
LVAZMNBKXWCIMF
|
8.2 | IC50 | 3 | — | |
MFQHDSGLLLJSPV
|
8.2 | IC50 | 3 | — | |
NHIRQUMDHFNSGY
|
8.2 | IC50 | 3 | — | |
OZAALIWIRMBCOR
|
8.2 | IC50 | 4 | — | |
RWNSOGBUKTYZJZ
|
8.2 | IC50 | 3 | — | |
YNQGEMKAJKCOIP
|
8.2 | IC50 | 3 | — | |
PRHPCWAJDWRBJW
|
8.1 | IC50 | 3 | — | |
FUGVOKHOINFPBY
|
8.1 | IC50 | 3 | — | |
GAXARIICIJOJOY
|
8.1 | IC50 | 3 | — | |
JAVVLMYHUYZZDN
|
8.1 | IC50 | 3 | — | |
MXHQJSWMMQETFE
|
8.1 | IC50 | 8 | — | |
RMTAUHCHXYNQOT
|
8.1 | IC50 | 3 | — | |
USPNCTNCYQFTGT
|
8.1 | IC50 | 3 | — | |
ANSIRGLMUHWNPB
|
8.1 | IC50 | 3 | — | |
DECHCVMZNFKMLE
|
8.1 | IC50 | 3 | — | |
DJNAAVCOMOYFNT
|
8.1 | IC50 | 3 | — | |
FVRMTRYCXIUJEB
|
8.1 | IC50 | 3 | — | |
FVRMTRYCXIUJEB
|
8.1 | IC50 | 3 | — | |
GHBOTNLUBMTSJO
|
8.1 | IC50 | 3 | — | |
HIRGJKYVLHTQTI
|
8.1 | IC50 | 3 | — | |
MGVBQZCURGNGQO
|
8.1 | IC50 | 3 | — | |
NGHKXECWEKEJAN
|
8.1 | Ki | 3 | — | |
UCSBUXYSZFPGSI
|
8.1 | IC50 | 3 | — | |
UJCZXEMKGRZREN
|
8.1 | IC50 | 5 | — | |
URLSXEUWUQRQEM
|
8.1 | IC50 | 5 | — | |
UUIYNZNVNQVZOT
|
8.1 | IC50 | 5 | — | |
VNFMQMVCRRHLOL
|
8.1 | IC50 | 3 | — | |
VNGYQBMDQMDALH
|
8.1 | Ki | 25 | — | |
CHFXZLZGCMQMBM
|
8.1 | IC50 | 3 | — | |
YZAQSGMOAYQDAV
|
8.1 | IC50 | 3 | — | |
IIFMWBFXGMFSOH
|
8.1 | IC50 | 3 | — |