Target Details
| UniProt AC | Q86V86 |
|---|---|
| Gene Symbol | PIM3 |
| Protein Name | Serine/threonine-protein kinase pim-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,417
- Clinical molecules 10
- Avg pChEMBL 8.16
Active Molecules (1,417)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WUTCYYSJWLOLPF
|
8.5 | IC50 | 3 | — | |
YKTHPBIEPMMOPM
|
8.5 | IC50 | 3 | — | |
YNWQVSDBNPDGBY
|
8.4 | IC50 | 3 | — | |
MILQRCUVJFKCQR
|
8.4 | Ki | 3 | — | |
MMOSRHUYBPJLSR
|
8.4 | IC50 | 3 | — | |
OSSMVZDTZQMDKR
|
8.4 | IC50 | 3 | — | |
RJYKOWGBWXBBBA
|
8.4 | IC50 | 3 | — | |
KKTIVBUXNOFPPA
|
8.4 | IC50 | 3 | — | |
LNIXAFUYUNLOOW
|
8.4 | Ki | 3 | — | |
BJWZYPUXMABVIE
|
8.4 | IC50 | 3 | — | |
BGFPXHMHXQXNPY
|
8.4 | IC50 | 3 | — | |
BKUXTVCORRDHGA
|
8.4 | IC50 | 3 | — | |
FRRLLRQAGKSVMU
|
8.4 | IC50 | 7 | — | |
GOFOMUKPTQCOQX
|
8.4 | Ki | 3 | — | |
GOYXKJXQXYESKZ
|
8.4 | IC50 | 3 | — | |
HWIDISMNBLRQNP
|
8.4 | IC50 | 3 | — | |
HWNZDLXOJIRFFD
|
8.4 | IC50 | 3 | — | |
JBHWJIFAFZAYFD
|
8.4 | IC50 | 2 | — | |
JSWXHRIKDWHCOW
|
8.4 | IC50 | 3 | — | |
LQASHUDUJOBHMP
|
8.4 | IC50 | 3 | — | |
LYAZTMOXEBYWIS
|
8.4 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
8.4 | Kd | 200 | — | |
PAWYDNPYJNAJHA
|
8.4 | IC50 | 3 | — | |
QVCLVTVRXGXXOR
|
8.4 | Ki | 4 | — | |
SCFVVTCJKWYEAW
|
8.4 | IC50 | 3 | — | |
SCFVVTCJKWYEAW
|
8.4 | IC50 | 3 | — | |
SDSSZBQMUURFEC
|
8.4 | IC50 | 3 | — | |
SKYIOLUXCWYHKN
|
8.4 | IC50 | 3 | — | |
SLGWCOFFSAFFES
|
8.4 | Ki | 3 | — | |
SNHNWCQKOINDPL
|
8.4 | IC50 | 3 | — | |
STWDLMHONRHMTF
|
8.4 | IC50 | 3 | — | |
VBJQFXDREPPTOL
|
8.4 | IC50 | 3 | — | |
VNHNIGCSETXKQL
|
8.4 | Ki | 2 | — | |
WIPBIZXEEPHOTH
|
8.4 | IC50 | 3 | — | |
WROQCXULSBZMCN
|
8.4 | IC50 | 3 | — | |
XDENGFSQWNBWJS
|
8.4 | IC50 | 3 | — | |
XQKKLBDDZJZNLU
|
8.4 | IC50 | 3 | — | |
YJGTXPJKAHYANC
|
8.4 | IC50 | 3 | — | |
YUGYQVSNIPXJJV
|
8.4 | IC50 | 3 | — | |
ZNTIFAHOYOIGGK
|
8.4 | IC50 | 3 | — | |
WUOXBBAOJFCZKX
|
8.4 | IC50 | 3 | — | |
FEIGOJWLHHRBHZ
|
8.4 | IC50 | 3 | — | |
JHCXRIDGVGVKMB
|
8.4 | IC50 | 3 | — | |
NBZYCEPNLRVSAP
|
8.4 | IC50 | 3 | — | |
SYEYZQUZNVVCNN
|
8.4 | IC50 | 3 | — | |
YGEIOFPNCMIFRQ
|
8.4 | IC50 | 3 | — | |
GWRLSNACWTZFNG
|
8.4 | IC50 | 3 | — | |
RXCHWYUVXYDNBW
|
8.4 | IC50 | 3 | — | |
WUOBKQMEZQEJEO
|
8.4 | IC50 | 3 | — | |
YTBQJCHZAHBGOV
|
8.4 | IC50 | 3 | — |