Target Details
| UniProt AC | Q86U86 |
|---|---|
| Gene Symbol | PBRM1 |
| Protein Name | Protein polybromo-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01426 (BAH) PF00439 (Bromodomain) PF00505 (HMG_box) |
Summary
- Multi-target molecules 53
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (53)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GSAKHYJGZSBABY
|
8.6 | IC50 | 3 | — | |
JISLSABSHWDDTJ
|
8.4 | IC50 | 3 | — | |
QMIHYQHNCMLKCV
|
8.3 | IC50 | 3 | — | |
VVYATDRFTFUUGA
|
8.3 | IC50 | 3 | — | |
HRPWASOMWDRLHQ
|
8.2 | IC50 | 3 | — | |
URAFMSDXCRQVKY
|
8.1 | IC50 | 3 | — | |
QGHVJDGMJOVMCR
|
8.0 | IC50 | 3 | — | |
FQZVWWGALUEODH
|
8.0 | Kd | 3 | — | |
AQTNUGRRZDRZIA
|
7.9 | Kd | 3 | — | |
SFMYKATXFFQSND
|
7.9 | IC50 | 3 | — | |
KXXHZDPNIIOTSH
|
7.8 | Kd | 3 | — | |
AFMDWCUFHCSFCR
|
7.8 | Kd | 4 | — | |
AKIDLWUESNUXNK
|
7.8 | IC50 | 3 | — | |
RNFAVDGGNIENKQ
|
7.8 | IC50 | 3 | — | |
FHRKRGDHMCCDEO
|
7.8 | IC50 | 3 | — | |
NCSVRIYOFWYLNA
|
7.8 | IC50 | 3 | — | |
HYFYBIOFAMANIC
|
7.7 | IC50 | 3 | — | |
JEKZPGPLMPQKGR
|
7.7 | IC50 | 3 | — | |
DTWXURVEXMCFCP
|
7.6 | IC50 | 3 | — | |
RJVQZTLPHCJXNB
|
7.6 | Kd | 3 | — | |
YRLBOSSSZSLHJB
|
7.6 | Kd | 4 | — | |
LTQBMPHICDLNOB
|
7.6 | IC50 | 3 | — | |
MBDFNLARUDVNEJ
|
7.6 | IC50 | 3 | — | |
SPSLNCYVKLGTKH
|
7.6 | IC50 | 3 | — | |
JZLOJEOBZZJRHN
|
7.6 | IC50 | 3 | — | |
SZKHGLTYXIDOFH
|
7.6 | Kd | 3 | — | |
COKXUIZUCWUEQS
|
7.5 | IC50 | 3 | — | |
LAMLMRYWDMUTPN
|
7.5 | IC50 | 3 | — | |
TWJZDPRYXHWSDF
|
7.5 | Kd | 3 | — | |
YIQNHNMFVVDQQU
|
7.5 | IC50 | 3 | — | |
CMJYPZQQLQOFCI
|
7.4 | Kd | 4 | — | |
BTCGLYACXJHVJC
|
7.4 | IC50 | 3 | — | |
NSAUQIQMBFHQRE
|
7.3 | IC50 | 3 | — | |
INAICWLVUAKEPB
|
7.3 | Kd | 4 | — | |
KZRXTHZVIAAZAP
|
7.3 | Kd | 3 | — | |
VZDXUFDLQRAMEG
|
7.3 | IC50 | 3 | — | |
KXXHZDPNIIOTSH
|
7.3 | Kd | 3 | — | |
SDAWPVIWTVUTCC
|
7.3 | Kd | 3 | — | |
NLFXZOJMKTYTIY
|
7.3 | Kd | 3 | — | |
IABGSEADKPXCRQ
|
7.2 | Kd | 2 | — | |
FHRKRGDHMCCDEO
|
7.0 | Kd | 3 | — | |
AAAQFGUYHFJNHI
|
7.0 | IC50 | 252 | — | |
ICVVDNFTMKQVQK
|
7.0 | IC50 | 3 | — | |
VLPRXFLUVHYBBT
|
6.9 | Kd | 3 | — | |
CMJYPZQQLQOFCI
|
6.9 | Kd | 3 | — | |
INAICWLVUAKEPB
|
6.8 | IC50 | 2 | — | |
VUGYKDOKOLKKRA
|
6.6 | Kd | 3 | — | |
SIWZRTOJDAJYHG
|
6.6 | IC50 | 3 | — | |
LTOWBWFTKOUSOO
|
6.6 | IC50 | 3 | — | |
DHDZFJQQXROKLC
|
6.5 | Kd | 3 | — |