Target Details
| UniProt AC | Q86U44 |
|---|---|
| Gene Symbol | METTL3 |
| Protein Name | N(6)-adenosine-methyltransferase catalytic subunit METTL3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05063 (MT-A70) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.47
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YJICMHRPAOFCRY
|
7.0 | IC50 | 2 | — | |
ZCFKJUKYINQBKY
|
7.0 | IC50 | 3 | — | |
ZCOJGQZPBAKOGD
|
7.0 | IC50 | 3 | — | |
ZLSHESUSBQPONM
|
7.0 | IC50 | 3 | — | |
DKFSYQKCEGWLCY
|
7.0 | IC50 | 2 | — | |
ICMRIVYUAVHOGM
|
7.0 | IC50 | 2 | — | |
LKGODYPZECUXPL
|
6.9 | IC50 | 2 | — | |
LMLFWEQIJTZXAJ
|
6.9 | IC50 | 2 | — | |
MCGSKRCIVZQMLU
|
6.9 | IC50 | 2 | — | |
WTVHEYXDICICGS
|
6.9 | IC50 | 2 | — | |
NQKRTKVWPQJYAH
|
6.8 | IC50 | 2 | — | |
SSEUTVLJEZDJNA
|
6.8 | IC50 | 2 | — | |
WUNVKARTCSOQRI
|
6.8 | IC50 | 2 | — | |
GHPDGAWBKYHSSO
|
6.7 | IC50 | 2 | — | |
HSUMIFOMDGDEEI
|
6.7 | IC50 | 2 | — | |
DKXCRAJRENEIRM
|
6.7 | IC50 | 2 | — | |
RTLJDTSKAYUCMC
|
6.7 | IC50 | 2 | — | |
FXNNSNRGNUOUKG
|
6.6 | IC50 | 2 | — | |
ODKRIBQJCPIBGJ
|
6.6 | IC50 | 2 | — | |
NMGYMKHSSFBFDP
|
6.6 | IC50 | 2 | — | |
IMOSBSGKJXQBOZ
|
6.6 | IC50 | 2 | — | |
PWYRDVXYAOGDNK
|
6.5 | IC50 | 2 | — | |
RJEWLHZZXYDBNT
|
6.5 | IC50 | 2 | — | |
UHMCBSCAUJSRCU
|
6.5 | IC50 | 2 | — | |
QDEZAWSGRHOJQM
|
6.5 | IC50 | 2 | — | |
HGXMRDNOWZGHFE
|
6.5 | IC50 | 2 | — | |
RAPWRVCEVCNOPC
|
6.5 | IC50 | 2 | — | |
WYXXBCJCGIHNFR
|
6.4 | IC50 | 2 | — | |
PWDAEZLLDYCGNZ
|
6.4 | IC50 | 2 | — | |
GSEZFABTMRQFRS
|
6.3 | IC50 | 2 | — | |
HTDDSGWGRCEXGP
|
6.3 | IC50 | 2 | — | |
XOOCXXDKKKMECD
|
6.3 | IC50 | 2 | — | |
PWMRWTBTFJIKMN
|
6.3 | IC50 | 2 | — | |
JWHLLJDYOCMKNH
|
6.3 | IC50 | 2 | — | |
ZPWPJARNYIVPFW
|
6.3 | IC50 | 2 | — | |
DSZUJZGHRPRNJW
|
6.3 | IC50 | 2 | — | |
AWEICSMJXXULJM
|
6.2 | IC50 | 2 | — | |
NFBCBNKSHLVTSS
|
6.2 | IC50 | 2 | — | |
ZJUKTBDSGOFHSH
|
6.2 | IC50 | 22 | — | |
BWCGOIFGMCWGMD
|
6.2 | IC50 | 2 | — | |
SDZSWRDDUPHAAY
|
6.2 | IC50 | 2 | — | |
TXPRNKKBKBMDAH
|
6.2 | IC50 | 2 | — | |
LLPUXUMPWGWUMW
|
6.1 | IC50 | 2 | — | |
BSVGKYJBSHYMPI
|
6.0 | IC50 | 2 | — | |
CSANZLJSAQBTMB
|
6.0 | IC50 | 2 | — | |
GBVXGNTZYNSJEA
|
6.0 | IC50 | 2 | — | |
GPZIVZOMXUPDAH
|
6.0 | IC50 | 2 | — | |
HCRXVBCEXCJJSV
|
6.0 | IC50 | 2 | — | |
IQAXJVBGIYHEKZ
|
6.0 | IC50 | 2 | — | |
KHBGXDWIVZWUNL
|
6.0 | IC50 | 2 | — |