Target Details
| UniProt AC | Q86U44 |
|---|---|
| Gene Symbol | METTL3 |
| Protein Name | N(6)-adenosine-methyltransferase catalytic subunit METTL3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05063 (MT-A70) |
Summary
- Multi-target molecules 309
- Clinical molecules 0
- Avg pChEMBL 7.47
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FAPUXZAAMCPCGI
|
7.8 | IC50 | 2 | — | |
IRIAVSJYFJXVGK
|
7.8 | IC50 | 2 | — | |
WEVJEDZAXXMEIM
|
7.8 | IC50 | 2 | — | |
YELNEYDBTGPVAO
|
7.7 | IC50 | 2 | — | |
TUIWZWXLGNLGBS
|
7.7 | IC50 | 2 | — | |
GTTUPSINADGZDV
|
7.7 | IC50 | 2 | — | |
NKMGGFLQYDFYHD
|
7.7 | IC50 | 2 | — | |
MEZCOHHISRKBRU
|
7.7 | IC50 | 2 | — | |
WJEVYKPGJXTIKS
|
7.6 | IC50 | 2 | — | |
NCIWOMQUDFJFDC
|
7.6 | IC50 | 2 | — | |
OOSMRIZGLAWLIZ
|
7.6 | IC50 | 2 | — | |
HGJWWKQXSAHGKQ
|
7.6 | IC50 | 2 | — | |
FKEUMAQBZXEVEA
|
7.6 | IC50 | 2 | — | |
GPXGOBHQOQMKDZ
|
7.6 | IC50 | 2 | — | |
DJSCPKOKUJKBJW
|
7.5 | IC50 | 2 | — | |
GDAACIHOBUCGGJ
|
7.5 | IC50 | 2 | — | |
FOXPVULNXFJYMT
|
7.5 | IC50 | 2 | — | |
LSPKIAXMFJWAHQ
|
7.4 | IC50 | 2 | — | |
FSMVOBUDPCUEOQ
|
7.4 | IC50 | 2 | — | |
XRUBPYKBZQFFLN
|
7.3 | IC50 | 2 | — | |
LOGVUKRPUBXIFN
|
7.3 | IC50 | 2 | — | |
RARBXVBXVAWUHA
|
7.2 | IC50 | 2 | — | |
FJLHJBBKTBGSDZ
|
7.2 | IC50 | 2 | — | |
NVOCCNITLYDGTN
|
7.2 | IC50 | 2 | — | |
VACQSTDQBDBCJL
|
7.2 | IC50 | 2 | — | |
BRBPDNLEJOXKOI
|
7.2 | IC50 | 2 | — | |
HUODOKZLAUIXJF
|
7.2 | IC50 | 2 | — | |
MRMZGBIWOUAIJS
|
7.2 | IC50 | 2 | — | |
OGFUDMMHTPTUCZ
|
7.1 | IC50 | 2 | — | |
ZVISABKROJHWSL
|
7.1 | IC50 | 2 | — | |
SHASDQUWJUXLDV
|
7.1 | IC50 | 2 | — | |
SXLRDIGWZWQBLL
|
7.0 | IC50 | 2 | — | |
AGYPZLZLPAXHPC
|
7.0 | IC50 | 2 | — | |
AHSCEIIJIDWUSO
|
7.0 | IC50 | 3 | — | |
ARQMZHUCEQVMBR
|
7.0 | IC50 | 3 | — | |
BBPXWJIFZIZQJN
|
7.0 | IC50 | 3 | — | |
BSCNZRRBABACDM
|
7.0 | IC50 | 3 | — | |
BTVPTMWTKQPMRW
|
7.0 | IC50 | 3 | — | |
CPJMLOLDZRVYHI
|
7.0 | IC50 | 3 | — | |
CZQDXGWPFGVYEA
|
7.0 | IC50 | 2 | — | |
DMTXVXQTQRVQHI
|
7.0 | IC50 | 3 | — | |
DRJLIJVRIGWPPF
|
7.0 | IC50 | 3 | — | |
DRJLIJVRIGWPPF
|
7.0 | IC50 | 3 | — | |
DWKQTUXGXSWCDD
|
7.0 | IC50 | 3 | — | |
FEAJNCPPXMPQES
|
7.0 | IC50 | 3 | — | |
FQCUFTGCWIMALT
|
7.0 | IC50 | 3 | — | |
FZMXQSIAXDAVST
|
7.0 | IC50 | 2 | — | |
GTDKKNHZRPOBLP
|
7.0 | IC50 | 3 | — | |
GVJMFHDJGPYKLA
|
7.0 | IC50 | 3 | — | |
HJXJQDDRWMMLCV
|
7.0 | IC50 | 3 | — |