Target Details
| UniProt AC | Q848S6 |
|---|---|
| Gene Symbol | bla |
| Protein Name | Carbapenem-hydrolyzing beta-lactamase KPC |
| Organism | Klebsiella oxytoca |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 7.05
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KOHUFVUIYUCFNG
|
8.7 | Ki | 4 | — | |
IUNQEXJRZWMEMG
|
7.7 | Ki | 2 | — | |
IOOWNWLVCOUUEX
|
7.2 | Ki | 2 | — | |
SDYHQCDQJPLOQK
|
6.8 | Ki | 2 | — | |
UKVXZBVYSYLEHH
|
6.5 | Ki | 2 | — | |
USZAGAREISWJDP
|
6.2 | IC50 | 7 | — | |
AXDYXEZTDRQFQK
|
6.1 | Ki | 2 | — |