Target Details
| UniProt AC | Q81R22 |
|---|---|
| Gene Symbol | dfrA |
| Protein Name | Dihydrofolate reductase |
| Organism | Bacillus anthracis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) |
Summary
- Multi-target molecules 13
- Clinical molecules 0
- Avg pChEMBL 6.56
Active Molecules (13)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBOZXECLQNJBKD
|
7.8 | IC50 | 16 | — | |
YGDVMSPWZQHNMB
|
7.3 | IC50 | 2 | — | |
RUQVXLIOJPKNCM
|
6.8 | Ki | 4 | — | |
OEYXETAXVXPYMF
|
6.4 | Ki | 3 | — | |
DGJGWMFHVPDAKM
|
6.4 | Ki | 4 | — | |
MRGVCWULZNEIIL
|
6.4 | Ki | 2 | — | |
WJIMEKODTQDGFJ
|
6.4 | IC50 | 4 | — | |
QKLZHVMWTSBUFL
|
6.4 | IC50 | 4 | — | |
LBQMRSNKEUNXMT
|
6.4 | IC50 | 4 | — | |
IEDVJHCEMCRBQM
|
6.3 | Ki | 7 | — | |
JPENSYBRTSIYGO
|
6.3 | IC50 | 5 | — | |
VPNXKXUNASBBLU
|
6.3 | IC50 | 3 | — | |
NNFDQABYXZBKRK
|
6.0 | IC50 | 4 | — |