Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
INZUGTGTHGBOFW
|
7.8 | IC50 | 2 | — | |
JRVAAZSLJJQIES
|
7.8 | IC50 | 2 | — | |
KBWNGLRCTYSSQQ
|
7.8 | IC50 | 2 | — | |
NBBLWTOHJFZTMU
|
7.8 | IC50 | 2 | — | |
UAKPLSPFKYUCEA
|
7.8 | IC50 | 2 | — | |
UQGLWKQYJVYZSD
|
7.8 | IC50 | 2 | — | |
FKTXCMVVZXVLFV
|
7.8 | IC50 | 2 | — | |
VJTGPVBZBWOCRZ
|
7.8 | IC50 | 2 | — | |
CZFFBEXEKNGXKS
|
7.8 | IC50 | 4 | — | |
LZJPQUXPORHTNN
|
7.8 | IC50 | 2 | — | |
NLISQTHJICPFKQ
|
7.8 | IC50 | 2 | — | |
OUOKKABEASKAHZ
|
7.8 | IC50 | 2 | — | |
UDWMEZOSHUGYOG
|
7.8 | IC50 | 2 | — | |
MMZRUVLLFMTCOG
|
7.8 | IC50 | 2 | — | |
XESKIKFUQNEPGO
|
7.8 | IC50 | 2 | — | |
ZVVUFFNOQHYLCA
|
7.8 | IC50 | 2 | — | |
DODMZNFPNFKNSU
|
7.8 | IC50 | 2 | — | |
GDDBKURUXLFLCG
|
7.8 | IC50 | 2 | — | |
HJTLTRSQUNLHAL
|
7.8 | IC50 | 2 | — | |
KMLKSQSEXABFBS
|
7.8 | IC50 | 2 | — | |
MSHIMSJOYGFYNB
|
7.8 | IC50 | 2 | — | |
NHCFEOHLENNJPQ
|
7.8 | IC50 | 2 | — | |
PWEVLUAHMYMYHE
|
7.8 | IC50 | 2 | — | |
QGXFBKLVCZDQRD
|
7.8 | IC50 | 2 | — | |
REFNAZZRMUJXTD
|
7.8 | IC50 | 2 | — | |
SRROGGHIEHJFQH
|
7.8 | IC50 | 2 | — | |
UINLNNHMBXVCDU
|
7.8 | IC50 | 2 | — | |
FPVPQIOUSAJQDM
|
7.7 | IC50 | 2 | — | |
MWPWGZXQCAMTQA
|
7.7 | IC50 | 3 | — | |
IKUFIINOCOGAOY
|
7.7 | IC50 | 2 | — | |
ITAODOQMELNLOA
|
7.7 | IC50 | 2 | — | |
JGNGTGUUSAINFD
|
7.7 | IC50 | 2 | — | |
ONPKMIYEKBFJSF
|
7.7 | IC50 | 2 | — | |
PEBWIPMJIWZNLD
|
7.7 | IC50 | 2 | — | |
RNJYHOYBLXEGDT
|
7.7 | IC50 | 2 | — | |
SRUNQRKISSFNSQ
|
7.7 | IC50 | 2 | — | |
AJGWMYJQISFUBH
|
7.7 | IC50 | 2 | — | |
AOKHOZKILWTAKY
|
7.7 | IC50 | 2 | — | |
AOVMSLZGYMUDKX
|
7.7 | IC50 | 2 | — | |
AWXUJSKCZCJLCA
|
7.7 | IC50 | 2 | — | |
AYYZVIZCPBKXCO
|
7.7 | IC50 | 2 | — | |
BGZBLIWCOTUAQD
|
7.7 | IC50 | 2 | — | |
DMTQWFCGBWIWPC
|
7.7 | IC50 | 2 | — | |
DWNWXQVKMRJASU
|
7.7 | IC50 | 2 | — | |
FBHOZTRRKYTTHS
|
7.7 | IC50 | 2 | — | |
FLPRWHQUZWATIH
|
7.7 | IC50 | 2 | — | |
FSFOUSUJEBSBEN
|
7.7 | IC50 | 2 | — | |
GLRLTCIJLBXDEU
|
7.7 | IC50 | 2 | — | |
HTCXQAIZGKXKOW
|
7.7 | IC50 | 2 | — | |
ICPPCODEZYGZTO
|
7.7 | IC50 | 2 | — |