Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NENPYTRHICXVCS
|
8.0 | IC50 | 3 | — | |
OKLYWXAJDGCACQ
|
8.0 | IC50 | 4 | — | |
PSMBVVQBAVEJQO
|
8.0 | IC50 | 2 | — | |
QBJQWIQAJVYVTJ
|
8.0 | IC50 | 2 | — | |
RWCACWKLMSUOFC
|
8.0 | IC50 | 2 | — | |
SLWYUJVCKLWTGV
|
8.0 | IC50 | 2 | — | |
TWWLJWGXKQAITK
|
8.0 | IC50 | 2 | — | |
UJZVTGOPYAKBIB
|
8.0 | IC50 | 2 | — | |
UMPCIKHDGHZMJR
|
8.0 | IC50 | 2 | — | |
WGLILLWPZIBWTQ
|
8.0 | IC50 | 2 | — | |
XWVTVSSPEHHYCE
|
8.0 | IC50 | 2 | — | |
YLSDEWQNSIAMQO
|
8.0 | IC50 | 3 | — | |
YMHFTOMTCCFRNK
|
8.0 | IC50 | 2 | — | |
YWYHIDAJZXGQKF
|
8.0 | IC50 | 2 | — | |
ZEVLDMFFBCKSHX
|
8.0 | IC50 | 2 | — | |
ZUIYPJQQZGBVLU
|
8.0 | IC50 | 2 | — | |
BWVZWKYMWWPRBX
|
8.0 | IC50 | 2 | — | |
CAWTUZMSASDZAZ
|
8.0 | IC50 | 2 | — | |
KYHZUFQVCKRYFE
|
8.0 | IC50 | 2 | — | |
QAWUWJFJRCHDON
|
8.0 | IC50 | 2 | — | |
QOZUICSVLJMIDW
|
8.0 | IC50 | 2 | — | |
WSCAFQQOJGOICA
|
8.0 | IC50 | 2 | — | |
ZEGNINTUGJBHLO
|
8.0 | IC50 | 2 | — | |
BMTUWFRODUAELZ
|
7.9 | IC50 | 2 | — | |
GAMTZJAHNULQKC
|
7.9 | IC50 | 2 | — | |
GBZVOYZIAPKRDQ
|
7.9 | IC50 | 2 | — | |
VIXSQLLJOWOFDW
|
7.9 | IC50 | 2 | — | |
YEFIJEXZAWLRFG
|
7.9 | IC50 | 2 | — | |
ZXDMPBVTUADOPS
|
7.9 | IC50 | 2 | — | |
VLXQXSPUFLVMKN
|
7.9 | IC50 | 3 | — | |
CHVSZADBLIGXGE
|
7.9 | IC50 | 2 | — | |
CMTZLJPHBPJAIR
|
7.9 | IC50 | 2 | — | |
CQJFSUBLVBRDAG
|
7.9 | IC50 | 2 | — | |
HTJZULVCICQELB
|
7.9 | IC50 | 2 | — | |
KCYDCUJLFCSMKX
|
7.9 | IC50 | 2 | — | |
YTQNZGHPUXHBMQ
|
7.9 | IC50 | 2 | — | |
RHWKPHLQXYSBKR
|
7.9 | IC50 | 3 | — | |
DYGQWEZNJAWTMH
|
7.9 | IC50 | 3 | — | |
GMRBRKNJPWLHBH
|
7.8 | IC50 | 2 | — | |
MICHNPFNQOVIOX
|
7.8 | IC50 | 2 | — | |
MMHODSINCYCTKD
|
7.8 | IC50 | 2 | — | |
OZQLTBGFEMVVPY
|
7.8 | IC50 | 2 | — | |
PBZCVULNNNFCSF
|
7.8 | IC50 | 2 | — | |
XRBIRQRZNGSARA
|
7.8 | IC50 | 2 | — | |
XRTUQGUSUCBJSA
|
7.8 | IC50 | 2 | — | |
JUZYLCPPVHEVSV
|
7.8 | IC50 | 2 | — | |
PPCMZJZCQJICAL
|
7.8 | IC50 | 2 | — | |
CZFFBEXEKNGXKS
|
7.8 | IC50 | 2 | — | |
DUQLQAPYMYISEO
|
7.8 | IC50 | 2 | — | |
INYVTIRVESMVAC
|
7.8 | IC50 | 2 | — |